SCHEMBL4746002

SCHEMBL4746002

CC(C)(C)OC(=O)Nc1cc(Br)cc2c1C(=O)N(Cc1ccc(F)cc1F)C2=O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 3/20 0.40
GRM5 P41594 3/20 0.38
AAK1 Q2M2I8 2/20 0.36
AKR1B10 O60218 1/20 0.35
AKR1A1 P14550 1/20 0.35
HSD17B10 Q99714 1/20 0.35
KCNQ4 P56696 1/20 0.35
KCNQ5 Q9NR82 1/20 0.35
PTGER1 P34995 2/20 0.34
ACHE P22303 4/20 0.34
RIPK3 Q9Y572 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4748502 0.83 IDO1 (0.41) GRM5
SCHEMBL4745710 0.81 KCNA5 (0.35) AKR1B1AAK1KCNQ4KCNQ5RIPK3
SCHEMBL4745826 0.81 KCNA5 (0.35) AKR1B1AAK1KCNQ4KCNQ5PTGER1
SCHEMBL4749155 0.79 AAK1 (0.36) AAK1KCNQ4KCNQ5
SCHEMBL4749154 0.79 AAK1 (0.36) AAK1KCNQ4KCNQ5
SCHEMBL4518262 0.75 AKR1B1 (0.45) AKR1B1AKR1B10AKR1A1ACHE
SCHEMBL4518252 0.74 AKR1B1 (0.48) AKR1B1GRM5AKR1B10AKR1A1PTGER1
SCHEMBL3750959 0.74 RORC (0.37) AAK1
SCHEMBL3750954 0.74 RORC (0.37) AAK1
SCHEMBL857284 0.69 HTT (0.55) KCNQ4KCNQ5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008124518-A1 OXO-DIHYDROISOINDOLE SULFONAMIDE COMPOUNDS AS MODULATORS OF THE CCK2 RECEPTOR JANSSEN PHARMACEUTICA N.V. (BE) 2008-10-16 WO disclosed