SCHEMBL4746032

SCHEMBL4746032

Nc1cc(Br)cc2c1C(=O)N(Cc1ccc(F)cc1F)C2

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 8/20 0.39
KDM4E B2RXH2 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CHRM1 P11229 1/20 0.36
AKR1B1 P15121 2/20 0.35
AKR1B10 O60218 1/20 0.35
AKR1A1 P14550 1/20 0.35
BDKRB1 P46663 1/20 0.35
CLPP Q16740 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4748978 0.81 P2RX7 (0.39) P2RX7KDM4ESMN1; SMN2CHRM1AKR1B1
SCHEMBL4518262 0.77 AKR1B1 (0.45) KDM4ESMN1; SMN2AKR1B1AKR1B10AKR1A1
SCHEMBL13952113 0.73 KDM4E (0.40) KDM4ESMN1; SMN2CHRM1
SCHEMBL15729520 0.73 BDKRB1 (0.44) KDM4ESMN1; SMN2BDKRB1
SCHEMBL2029868 0.72 P2RX7 (0.46) P2RX7KDM4EBDKRB1
SCHEMBL4748815 0.72 HSD11B1 (0.39)
SCHEMBL2028436 0.72 BDKRB1 (0.58) KDM4ESMN1; SMN2CHRM1BDKRB1
SCHEMBL29303348 0.72 GRM2 (0.47) AKR1B1BDKRB1
SCHEMBL15729563 0.71 BDKRB1 (0.48) P2RX7KDM4ESMN1; SMN2BDKRB1
SCHEMBL2020826 0.70 MAPK1 (0.42) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008124518-A1 OXO-DIHYDROISOINDOLE SULFONAMIDE COMPOUNDS AS MODULATORS OF THE CCK2 RECEPTOR JANSSEN PHARMACEUTICA N.V. (BE) 2008-10-16 WO claimed
WO-2008124518-A1 OXO-DIHYDROISOINDOLE SULFONAMIDE COMPOUNDS AS MODULATORS OF THE CCK2 RECEPTOR JANSSEN PHARMACEUTICA N.V. (BE) 2008-10-16 WO disclosed