SCHEMBL4746574

SCHEMBL4746574

Cc1oc(-c2ccc(C(F)(F)F)cc2)nc1COc1ccc(CN2CCCC2C(=O)O)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
KDM4E B2RXH2 1/20 0.49
PPARG P37231 9/20 0.48
PPARA Q07869 8/20 0.48
CD274 Q9NZQ7 1/20 0.48
PPARD Q03181 3/20 0.48
FFAR1 O14842 1/20 0.48
CYP2C9 P11712 1/20 0.48
KCNH2 Q12809 1/20 0.48
PTPN1 P18031 1/20 0.47
NPSR1 Q6W5P4 1/20 0.46
SPHK2 Q9NRA0 1/20 0.46
SPHK1 Q9NYA1 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
S1PR1 P21453 1/20 0.45
S1PR3 Q99500 1/20 0.45
S1PR5 Q9H228 1/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4748026 1.00 ALDH1A1 (0.49) ALDH1A1KDM4EPPARGPPARACD274
SCHEMBL4748235 1.00 ALDH1A1 (0.49) ALDH1A1KDM4EPPARGPPARACD274
SCHEMBL4744570 0.98 KDM4E (0.52) ALDH1A1KDM4EPPARGPPARACD274
SCHEMBL4744563 0.98 KDM4E (0.52) ALDH1A1KDM4EPPARGPPARACD274
SCHEMBL4744028 0.93 PPARG (0.56) PPARGPPARAPPARDCYP2C9KCNH2
SCHEMBL4748056 0.93 PPARG (0.56) PPARGPPARAPPARDCYP2C9KCNH2
SCHEMBL4744558 0.92 ALDH1A1 (0.51) ALDH1A1KDM4EPPARGPPARAPPARD
SCHEMBL4788139 0.92 ALDH1A1 (0.51) ALDH1A1KDM4EPPARGPPARAPPARD
SCHEMBL4744562 0.92 ALDH1A1 (0.51) ALDH1A1KDM4EPPARGPPARAPPARD
SCHEMBL4743758 0.91 PPARG (0.57) PPARGPPARACD274FFAR1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008117982-A1 HETEROCYCLIC CARBOXYLIC ACID DERIVATIVES AND PHARMACEUTICAL COMPOSITION FOR INHIBITING LIPID ACCUMULATION CONTAINING SAME CRYSTAL GENOMICS, INC. (KR) 2008-10-02 WO claimed
WO-2008117982-A1 HETEROCYCLIC CARBOXYLIC ACID DERIVATIVES AND PHARMACEUTICAL COMPOSITION FOR INHIBITING LIPID ACCUMULATION CONTAINING SAME CRYSTAL GENOMICS, INC. (KR) 2008-10-02 WO disclosed