SCHEMBL4747170

SCHEMBL4747170

COc1cccc(-c2nc(C)cc3c2C(=O)OCC3)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.45
ADORA1 P30542 1/20 0.45
KDM4E B2RXH2 2/20 0.41
HSD17B10 Q99714 2/20 0.41
LMNA P02545 1/20 0.41
ALOX5 P09917 1/20 0.41
GAA P10253 1/20 0.40
PFKFB3 Q16875 1/20 0.39
BRD4 O60885 1/20 0.39
NOTUM Q6P988 1/20 0.39
PDE7A Q13946 1/20 0.39
PDE3A Q14432 1/20 0.39
PDE10A Q9Y233 1/20 0.39
HPGD P15428 4/20 0.39
ALDH1A1 P00352 2/20 0.39
KMT2A Q03164 2/20 0.39
F2 P00734 1/20 0.39
TP53 P04637 1/20 0.39
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4065342 0.83 L3MBTL1 (0.45) ADORA2AADORA1KDM4EHSD17B10LMNA
SCHEMBL4749649 0.81 PFKFB3 (0.43) ADORA2AADORA1KDM4EHSD17B10ALOX5
SCHEMBL4072063 0.78 MAPK1 (0.40) ADORA2AADORA1KDM4EHSD17B10LMNA
SCHEMBL4072395 0.78 NPC1 (0.39) ADORA2AADORA1KDM4EHSD17B10LMNA
SCHEMBL11485963 0.76 HTR1A (0.45) ADORA2AADORA1KDM4ELMNAALOX5
SCHEMBL4070664 0.75 KDM4E (0.41) KDM4EHSD17B10LMNAGAAHPGD
SCHEMBL4074599 0.75 KDM4E (0.40) ADORA2AADORA1KDM4EHSD17B10LMNA
SCHEMBL4070926 0.73 CYP1A2 (0.43) KDM4EHSD17B10LMNAGAAHPGD
SCHEMBL4251098 0.72 ADORA2A (0.35) ADORA2AADORA1KDM4EHSD17B10LMNA
SCHEMBL4070385 0.72 KDM4E (0.42) ADORA2AKDM4EHSD17B10GAAPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123756-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTON TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed