SCHEMBL474794

SCHEMBL474794

O=C(O)Oc1ccc(-c2cc(Cl)c(C[C@@H]3CCN(C4CCC(F)(F)CC4)C3=O)c(Cl)c2)cc1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 4/20 0.36
PARP1 P09874 4/20 0.33
ROCK2 O75116 3/20 0.33
CYP2D6 P10635 1/20 0.31
CYP2B6 P20813 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
CHRNA3 P32297 1/20 0.31
FFAR4 Q5NUL3 1/20 0.30
KCNJ6 P48051 1/20 0.30
KCNJ5 P48544 1/20 0.30
KCNJ3 P48549 1/20 0.30
SCN9A Q15858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474638 0.90 ROCK2 (0.33) HSD11B1PARP1ROCK2FFAR4KCNJ6
SCHEMBL474792 0.89 HSD11B1 (0.38) HSD11B1PARP1ROCK2CYP2D6CYP2B6
SCHEMBL3878885 0.88 HSD11B1 (0.49) HSD11B1
SCHEMBL474673 0.87 HSD11B1 (0.39) HSD11B1PARP1ROCK2CYP2D6CYP2B6
SCHEMBL474718 0.87 HSD11B1 (0.39) HSD11B1PARP1ROCK2KCNJ6KCNJ5
SCHEMBL474719 0.87 HSD11B1 (0.39) HSD11B1PARP1ROCK2KCNJ6KCNJ5
SCHEMBL474674 0.87 HSD11B1 (0.39) HSD11B1PARP1ROCK2CYP2D6CYP2B6
SCHEMBL474851 0.86 AKR1C2 (0.38) HSD11B1ROCK2FFAR4SCN9A
SCHEMBL13897773 0.86 HSD11B1 (0.35) HSD11B1PARP1ROCK2CYP2D6CYP2B6
SCHEMBL474642 0.86 AKR1C2 (0.38) HSD11B1ROCK2FFAR4SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049475-B1 CYCLOHEXYL SUBSTITUTED PYRROLIDINONES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE 1 LILLY CO ELI (US) 2012-02-01 EP claimed