SCHEMBL4748346

SCHEMBL4748346

Nc1ncc(-c2ccc3c(c2)NC(=O)CS3)c(N)n1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DHFR P00374 5/20 0.46
HTT P42858 2/20 0.44
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
PDE3B Q13370 3/20 0.40
PDE3A Q14432 3/20 0.40
MAOA P21397 2/20 0.39
MAOB P27338 2/20 0.39
EPHX2 P34913 1/20 0.39
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL395053 0.71 HTT (0.59) HTTCYP11B1CYP11B2NPC1RAB9A
SCHEMBL4258367 0.70 HTT (0.59) HTTCYP11B1CYP11B2NPC1ALDH1A1
SCHEMBL30648402 0.69 CYP11B1 (0.49) HTTCYP11B1CYP11B2NPC1RAB9A
SCHEMBL1723432 0.69 DHFR (0.44) DHFRALDH1A1
SCHEMBL4475827 0.68 DHFR (0.46) DHFRCYP11B1CYP11B2ALDH1A1MAPT
SCHEMBL29114864 0.68 DHFR (0.51) DHFR
SCHEMBL30648377 0.68 EPHX2 (0.47) HTTCYP11B1CYP11B2NPC1RAB9A
SCHEMBL30648398 0.68 KIF11 (0.46) HTTCYP11B1CYP11B2NPC1RAB9A
SCHEMBL9732854 0.67 PDE3B (0.82) HTTCYP11B1CYP11B2ALDH1A1LMNA
SCHEMBL3956743 0.67 PDE3B (0.50) DHFRPDE3BPDE3AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008118823-A2 COMPOSITIONS AND METHODS FOR INHIBITION OF THE JAK PATHWAY RIGEL PHARMACEUTICALS, INC. (US) 2008-10-02 WO disclosed