SCHEMBL4748624

SCHEMBL4748624

[AsH2]CCc1cccc(Br)c1

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.63
IDO1 P14902 2/20 0.50
AGXT P21549 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
MAOB P27338 2/20 0.47
SIGMAR1 Q99720 1/20 0.45
GPR84 Q9NQS5 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4399626 0.85 TAAR1 (0.74) TAAR1IDO1AGXTSMN1; SMN2TDP1
SCHEMBL4544274 0.81
SCHEMBL5240585 0.81 TAAR1 (0.68) TAAR1IDO1AGXTSMN1; SMN2TDP1
SCHEMBL19524669 0.79 TAAR1 (0.65) TAAR1IDO1AGXTSMN1; SMN2TDP1
SCHEMBL705920 0.79 TAAR1 (0.65) TAAR1IDO1AGXTSMN1; SMN2TDP1
SCHEMBL9660784 0.79 TAAR1 (0.65) TAAR1IDO1AGXTTDP1MAOB
SCHEMBL30688447 0.79 TAAR1 (0.65) TAAR1IDO1AGXTSMN1; SMN2TDP1
SCHEMBL1646500 0.77 TAAR1 (0.63) TAAR1IDO1AGXTSMN1; SMN2TDP1
SCHEMBL1513555 0.77 TAAR1 (0.63) TAAR1IDO1AGXTSMN1; SMN2TDP1
SCHEMBL235748 0.77 TAAR1 (1.00) TAAR1IDO1AGXTSMN1; SMN2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966163-A1 PYRIMIDINE DERIVATIVES USEFUL AS INHIBITORS OF PKC-THETA Boehringer Ingelheim International GmbH (DE) 2008-09-10 EP disclosed
WO-2007076247-A1 PYRIMIDINE DERIVATIVES USEFUL AS INHIBITORS OF PKC-THETA BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-07-05 WO disclosed