SCHEMBL4748705

SCHEMBL4748705

O=C(O)c1ccc2nc(NCCN3CCOCC3)sc2c1

nearest known ligand 0.60

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CASR P41180 1/20 0.60
NOS3 P29474 2/20 0.56
NOS1 P29475 2/20 0.56
NOS2 P35228 1/20 0.56
CSNK2A1 P68400 1/20 0.56
HSD17B10 Q99714 2/20 0.55
IDO1 P14902 1/20 0.53
HTT P42858 2/20 0.52
CLK1 P49759 2/20 0.52
KMT2A Q03164 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
MEN1 O00255 1/20 0.52
POLB P06746 1/20 0.52
ALDH1A1 P00352 1/20 0.52
MAPT P10636 1/20 0.52
ABL1 P00519 2/20 0.52
AURKB Q96GD4 3/20 0.50
MAP3K8 P41279 1/20 0.50
MET P08581 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5216603 0.82 NOS3 (0.60) NOS3NOS1NOS2IDO1HTT
SCHEMBL22639912 0.82 HTT (0.64) CASRNOS3NOS1NOS2IDO1
SCHEMBL5212987 0.80 ALDH1A1 (0.68) NOS3NOS1NOS2IDO1KMT2A
SCHEMBL22639860 0.79 KMT2A (0.66) CASRNOS3NOS1NOS2IDO1
SCHEMBL8350666 0.78 AURKB (0.78) AURKB
SCHEMBL6919054 0.77 AURKB (0.77) AURKB
SCHEMBL22639710 0.77 IDO1 (0.56) NOS3NOS1NOS2HSD17B10IDO1
SCHEMBL22640029 0.76 MET (0.54) CASRNOS3NOS1NOS2IDO1
SCHEMBL19921646 0.75 HSD17B10 (0.60) HSD17B10SMN1; SMN2POLBALDH1A1MAPT
SCHEMBL613934 0.74 ABL1 (0.69) HTTCLK1KMT2ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008124393-A1 BENZOTHIAZOLE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS IRM LLC (BM) 2008-10-16 WO disclosed