SCHEMBL4748907

SCHEMBL4748907

C=CCc1cc(NCS(=O)(=O)C(C)C)cc(C(=O)O)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.34
AKR1C2 P52895 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
FFAR1 O14842 1/20 0.33
PTGS2 P35354 1/20 0.33
KDM4E B2RXH2 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
MAPT P10636 1/20 0.32
PPARA Q07869 1/20 0.32
F2 P00734 1/20 0.32
F10 P00742 1/20 0.32
PLG P00747 1/20 0.32
F7 P08709 1/20 0.32
F3 P13726 1/20 0.32
ALDH1A1 P00352 1/20 0.31
TDP1 Q9NUW8 2/20 0.30
CYP3A4 P08684 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4751788 0.86 AKR1C3 (0.36) AKR1C3AKR1C2MEN1KMT2AFFAR1
SCHEMBL5831309 0.72 XDH (0.41) AKR1C3AKR1C2MEN1KMT2AKDM4E
SCHEMBL11786434 0.72 XDH (0.41) AKR1C3AKR1C2MEN1KMT2AKDM4E
SCHEMBL4748909 0.71 BACE1 (0.36) AKR1C3AKR1C2MEN1KMT2APTGS2
SCHEMBL4751790 0.66 BACE1 (0.36) AKR1C3AKR1C2MAPT
SCHEMBL1176840 0.66 POLB (0.39) AKR1C3AKR1C2MEN1KMT2AKDM4E
SCHEMBL10633163 0.65 MAPT (0.48) MEN1KMT2AKDM4ENPC1RAB9A
SCHEMBL1176614 0.65 ALDH1A1 (0.45) AKR1C3AKR1C2MEN1KMT2APTGS2
SCHEMBL18614934 0.62 MRGPRX4 (0.49) AKR1C3AKR1C2PPARA
SCHEMBL22017029 0.62 XDH (0.37) AKR1C3AKR1C2MEN1KMT2APTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008135488-A1 ASPARTYL PROTEASE INHIBITORS MEDIVIR AB (SE) 2008-11-13 WO disclosed