SCHEMBL4748909

SCHEMBL4748909

C=CCc1cc(C(=O)O)cc(N(C)S(=O)(=O)C(C)C)c1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 3/20 0.36
BACE2 Q9Y5Z0 1/20 0.36
PTGS2 P35354 1/20 0.33
MRGPRX4 Q96LA9 1/20 0.33
RXRA P19793 3/20 0.32
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
MAPT P10636 1/20 0.32
NR4A2 P43354 2/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
CYP3A4 P08684 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
TAS2R14 Q9NYV8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4751790 0.85 BACE1 (0.36) BACE1MRGPRX4RXRAAKR1C3AKR1C2
SCHEMBL7946697 0.75 BACE1 (0.34) BACE1RXRANR4A2
SCHEMBL11786434 0.73 XDH (0.41) AKR1C3AKR1C2MAPTMEN1KMT2A
SCHEMBL5831309 0.73 XDH (0.41) AKR1C3AKR1C2MAPTMEN1KMT2A
SCHEMBL4748907 0.71 AKR1C3 (0.34) PTGS2AKR1C3AKR1C2MAPTMEN1
SCHEMBL21104531 0.70 KMT2A (0.46) MAPTMEN1KMT2AALDH1A1TAS2R14
SCHEMBL8155821 0.68 BACE1 (0.41) BACE1
SCHEMBL1176840 0.67 POLB (0.39) MRGPRX4AKR1C3AKR1C2MAPTMEN1
SCHEMBL10633163 0.66 MAPT (0.48) MRGPRX4RXRAMAPTMEN1KMT2A
SCHEMBL4751788 0.66 AKR1C3 (0.36) AKR1C3AKR1C2MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008135488-A1 ASPARTYL PROTEASE INHIBITORS MEDIVIR AB (SE) 2008-11-13 WO disclosed