SCHEMBL4748990

SCHEMBL4748990

Cc1ccc2[nH]c(=O)n(C3CCNC3)c2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 3/20 0.58
CHRM2 P08172 2/20 0.58
CHRM4 P08173 1/20 0.58
CHRM5 P08912 1/20 0.58
CHRM3 P20309 1/20 0.58
KCNH2 Q12809 1/20 0.58
DAO P14920 1/20 0.49
OPRM1 P35372 8/20 0.48
OPRD1 P41143 3/20 0.48
OPRK1 P41145 3/20 0.48
CACNA1F O60840 2/20 0.48
ADRA1D P25100 2/20 0.48
HTR7 P34969 2/20 0.48
ADRA1A P35348 2/20 0.48
ADRA1B P35368 2/20 0.48
OPRL1 P41146 2/20 0.48
CACNA1D Q01668 2/20 0.48
CACNA1S Q13698 2/20 0.48
CACNA1C Q13936 2/20 0.48
PGR P06401 8/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL603514 0.92 CHRM1 (0.64) CHRM1CHRM2CHRM4CHRM5CHRM3
Hydrochloric Acid SCHEMBL4635789 0.90 CHRM1 (0.62) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL14365466 0.90 CHRM1 (0.70) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL14041660 0.86 CHRM1 (0.49) CHRM1CHRM2CHRM4CHRM5CHRM3
Hydrochloric Acid SCHEMBL4747177 0.85 CHRM1 (0.48) CHRM1CHRM2CHRM4CHRM5CHRM3
Trifluoroacetic Acid SCHEMBL15575285 0.82 CHRM1 (0.54) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL2636696 0.82 PGR (0.52) OPRM1PGRTNKS
SCHEMBL14041567 0.82 CHRM1 (0.56) CHRM1CHRM2CHRM4CHRM5CHRM3
SCHEMBL2636697 0.82 PGR (0.52) OPRM1PGRTNKS
SCHEMBL1760904 0.81 OPRM1 (0.57) CHRM1CHRM2CHRM4CHRM5CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008119712-A1 BENZOIMIDAZOLE DERIVATIVES WHICH HAVE ACTIVITY AT M1 RECEPTOR AND THEIR USES IN MEDICINE GLAXO GROUP LIMITED (GB) 2008-10-09 WO disclosed
WO-2008119712-A1 BENZOIMIDAZOLE DERIVATIVES WHICH HAVE ACTIVITY AT M1 RECEPTOR AND THEIR USES IN MEDICINE GLAXO GROUP LIMITED (GB) 2008-10-09 WO disclosed