SCHEMBL4749176

SCHEMBL4749176

O=C1CN(Cc2ccc(F)cc2)CCN1C[C@H]1CO1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.42
RAB9A P51151 1/20 0.42
ALDH1A1 P00352 1/20 0.41
POLB P06746 1/20 0.41
DRD4 P21917 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ATM Q13315 1/20 0.39
MAPT P10636 1/20 0.39
CLPP Q16740 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4752585 1.00 MCHR1 (0.42) MCHR1RAB9AALDH1A1POLBDRD4
SCHEMBL4751233 0.88 SIGMAR1 (0.43) MCHR1ALDH1A1DRD4MEN1KMT2A
SCHEMBL4751231 0.88 SIGMAR1 (0.43) MCHR1ALDH1A1DRD4MEN1KMT2A
SCHEMBL4751907 0.88 SIGMAR1 (0.43) MCHR1ALDH1A1DRD4MEN1KMT2A
SCHEMBL608348 0.80 MAPT (0.50) DRD4MEN1KMT2AATMMAPT
SCHEMBL4788151 0.76 SIGMAR1 (0.45) RAB9AALDH1A1DRD4MEN1KMT2A
SCHEMBL4748954 0.76 SIGMAR1 (0.45) RAB9AALDH1A1DRD4MEN1KMT2A
SCHEMBL23995201 0.73 ALDH1A1 (0.50) MCHR1RAB9AALDH1A1POLB
SCHEMBL5055491 0.69 APP (0.54) RAB9ADRD4MEN1KMT2AMAPT
SCHEMBL8117468 0.69 MAPT (0.67) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008136754-A1 NOVEL BENZYL - 2 -OXO-PIPERAZINYL/ 7-OXO/5-OXA- [1,4] DIAZEPANYL/ 2 -OXO- TETRAHYDROPYRIMIDINYL DERIVATIVES ASTRAZENECA AB (SE) 2008-11-13 WO disclosed
WO-2008136754-A1 NOVEL BENZYL - 2 -OXO-PIPERAZINYL/ 7-OXO/5-OXA- [1,4] DIAZEPANYL/ 2 -OXO- TETRAHYDROPYRIMIDINYL DERIVATIVES ASTRAZENECA AB (SE) 2008-11-13 WO disclosed