SCHEMBL4749586

SCHEMBL4749586

CCCc1nc(N)cc2c1C(=O)OCC2

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.35
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
GAA P10253 1/20 0.32
BACE1 P56817 1/20 0.31
HEXA P06865 1/20 0.31
HEXB P07686 1/20 0.31
DRD2 P14416 1/20 0.30
DRD3 P35462 1/20 0.30
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4808073 0.89 DYRK1A (0.39) DYRK1AGAAHEXAHEXBMAOA
SCHEMBL4064490 0.83 GLP1R (0.34) HEXAHEXBDRD2DRD3MAOA
SCHEMBL4749400 0.83 MAOA (0.35) GAADRD2DRD3MAOAMAOB
Hydrochloric Acid SCHEMBL4250086 0.82 MAOA (0.35) GAADRD2DRD3MAOAMAOB
SCHEMBL4749114 0.78 HRH4 (0.33) GAADRD2DRD3
SCHEMBL4072001 0.78 BACE1 (0.40) NOS3NOS1NOS2GAABACE1
SCHEMBL4746125 0.77 KDM4E (0.42) GAA
SCHEMBL4746139 0.77 ATM (0.34) GAA
SCHEMBL4245511 0.76 MAPT (0.32)
SCHEMBL4749246 0.74 DYRK1A (0.36) DYRK1ANOS3NOS1NOS2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123756-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTON TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed