SCHEMBL4749765

SCHEMBL4749765

NC(Cc1ccccc1)C(O)CNC1CC2CCC1C2

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
F2 P00734 2/20 0.40
CSNK1E P49674 1/20 0.39
LTA4H P09960 1/20 0.38
ALDH1A1 P00352 1/20 0.38
EPHX2 P34913 1/20 0.38
HSD17B10 Q99714 1/20 0.37
EPHX1 P07099 1/20 0.36
KCNJ6 P48051 1/20 0.35
KCNJ5 P48544 1/20 0.35
KCNJ3 P48549 1/20 0.35
DPP4 P27487 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4749760 1.00 HPGD (0.41) HPGDSMN1; SMN2F2CSNK1ELTA4H
Hydrochloric Acid SCHEMBL5222193 0.99 HPGD (0.40) HPGDSMN1; SMN2F2CSNK1ELTA4H
SCHEMBL4692382 0.81 EPHX2 (0.43) SMN1; SMN2F2CSNK1EEPHX2EPHX1
Hydrochloric Acid SCHEMBL5223403 0.80 EPHX2 (0.42) SMN1; SMN2F2CSNK1EEPHX2EPHX1
SCHEMBL4042402 0.78 REN (0.47) HPGDSMN1; SMN2ALDH1A1EPHX2HSD17B10
SCHEMBL14253003 0.78 GRIN2B (0.48) F2CSNK1EEPHX1
SCHEMBL5805296 0.78 GRIN2B (0.48) F2CSNK1EEPHX1
SCHEMBL4047960 0.78 GRIN2B (0.48) F2CSNK1EEPHX1
Hydrochloric Acid SCHEMBL6111346 0.77 GRIN2B (0.47) F2CSNK1EEPHX1
SCHEMBL5225345 0.77 KLK5 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1692143-B1 TRICYCLIC INDOLE HYDROXYETHYLAMINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2008-11-12 EP disclosed