SCHEMBL4750347

SCHEMBL4750347

Cc1cc(-c2c(C)nc(C)c3c2CCOC3=O)cc(C)c1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 5/20 0.48
MAOB P27338 2/20 0.48
BRD4 O60885 6/20 0.37
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
BRD2 P25440 1/20 0.33
NUAK1 O60285 1/20 0.33
IGF1R P08069 1/20 0.33
MET P08581 1/20 0.33
PIM1 P11309 1/20 0.33
SRC P12931 1/20 0.33
AXL P30530 1/20 0.33
AKT1 P31749 1/20 0.33
KDR P35968 1/20 0.33
NEK2 P51955 1/20 0.33
PLK1 P53350 1/20 0.33
PTK2 Q05397 1/20 0.33
PKN1 Q16512 1/20 0.33
AURKB Q96GD4 1/20 0.33
NEK6 Q9HC98 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4075462 0.75 MAOA (0.48) MAOAMAOBBRD4BRD2PTGS1
SCHEMBL4075636 0.69 MAOA (0.41) MAOAMAOBBRD4BRD2ALOX5
SCHEMBL4072428 0.69 MAOA (0.43) MAOAMAOBNUAK1IGF1RMET
Hydrochloric Acid SCHEMBL4073845 0.68 MAOA (0.42) MAOAMAOBALOX5PTGS1PTGS2
SCHEMBL30487613 0.65 MAOA (1.00) MAOAMAOBBRD4NUAK1IGF1R
SCHEMBL4063497 0.65 KDM4E (0.44) MAOAMAOBBRD4
SCHEMBL4749025 0.63 PIK3CA (0.39) MAOAMAOB
SCHEMBL4066514 0.63 GAA (0.43) MAOAMAOBNUAK1IGF1RMET
SCHEMBL10930504 0.63 ALOX5 (0.67) SRCALOX5PTGS1PTGS2CYP2C9
SCHEMBL4067976 0.63 MAOA (0.40) MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123756-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTON TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed
WO-2008123756-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTON TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO disclosed