SCHEMBL4749025

SCHEMBL4749025

Cc1nc(-c2cccc(O)c2)cc2c1C(=O)OCC2

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 8/20 0.39
MAOA P21397 2/20 0.38
MAOB P27338 2/20 0.38
HSD17B1 P14061 2/20 0.38
HSD17B2 P37059 2/20 0.38
PFKFB3 Q16875 1/20 0.38
PIK3R1 P27986 1/20 0.37
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
AKR1C1 Q04828 1/20 0.37
PIK3CD O00329 2/20 0.36
ABL1 P00519 1/20 0.36
PDE4B Q07343 1/20 0.36
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
FYN P06241 1/20 0.35
PRF1 P14222 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4066864 0.85 ALDH1A1 (0.39) MAOAMAOBPDE4B
SCHEMBL4749649 0.83 PFKFB3 (0.43) MAOBPFKFB3PDE4B
SCHEMBL4481191 0.79 ALDH1A1 (0.46)
SCHEMBL4073028 0.78 APP (0.36) MAOAMAOB
SCHEMBL4750253 0.78 BRD4 (0.46)
SCHEMBL4072428 0.77 MAOA (0.43) MAOAMAOB
Hydrochloric Acid SCHEMBL4073845 0.76 MAOA (0.42) MAOAMAOB
SCHEMBL4067545 0.75 PDE4B (0.37) MAOAMAOBPDE4B
SCHEMBL4063729 0.74 PDE10A (0.38)
Hydrochloric Acid SCHEMBL4247459 0.74 PDE4B (0.36) MAOAMAOBPDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123756-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTON TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed