SCHEMBL4750651

SCHEMBL4750651

COc1ccc(-n2ccc3cc(-c4ccccc4)nc(C)c3c2=O)cc1OC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.43
TSHR P16473 2/20 0.43
MAPK1 P28482 2/20 0.43
HSD17B10 Q99714 2/20 0.43
USP2 O75604 1/20 0.43
HTT P42858 1/20 0.43
ATM Q13315 1/20 0.43
EGFR P00533 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
ADORA1 P30542 1/20 0.42
MAPT P10636 5/20 0.42
GAA P10253 2/20 0.42
THRB P10828 1/20 0.42
MCHR1 Q99705 2/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4747261 0.89 EGFR (0.46) ALDH1A1MEN1KMT2AKDM4EMAPK1
SCHEMBL4747315 0.85 EGFR (0.49) ALDH1A1MEN1KMT2AKDM4EEGFR
SCHEMBL5816238 0.81 ALDH1A1 (0.40) ALDH1A1KDM4EMAPK1HTTL3MBTL1
SCHEMBL4747892 0.80 ALDH1A1 (0.42) ALDH1A1MEN1KMT2AKDM4EHPGD
SCHEMBL4747889 0.79 ALDH1A1 (0.40) ALDH1A1MEN1KMT2AKDM4EHPGD
SCHEMBL4750620 0.75 RAD51 (0.40) ALDH1A1MEN1KMT2AEGFRL3MBTL1
SCHEMBL4248495 0.74 ALDH1A1 (0.47) ALDH1A1MEN1KMT2AKDM4EHPGD
SCHEMBL4747281 0.72 EGFR (0.46) ALDH1A1MEN1KMT2AHSD17B10EGFR
SCHEMBL4750229 0.71 CYP19A1 (0.45) ALDH1A1KDM4ETSHRMAPK1MAPT
SCHEMBL4750005 0.71 RAD51 (0.39) ALDH1A1MEN1KMT2AKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008123755-A1 A PHARMACEUTICAL COMPOSITIONS CONTAINING LACTAM TYPE PYRIDINE DERIVATIVES AS AN EFFECTIVE INGREDIENT FOR THE PREVENTION AND TREATMENT OF ISCHEMIA SK CHEMICALS CO., LTD. (KR) 2008-10-16 WO claimed
WO-2006112666-A1 PYRIDINE DERIVATIVES, METHODS OF THEIR PREPARATIONS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SK CHEMICALS CO., LTD. (KR) 2006-10-26 WO claimed
WO-2006112666-A1 PYRIDINE DERIVATIVES, METHODS OF THEIR PREPARATIONS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME SK CHEMICALS CO., LTD. (KR) 2006-10-26 WO disclosed