SCHEMBL4751748

SCHEMBL4751748

OCc1cccc(Nc2ccnc3cc(Cl)ccc23)c1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.70
NR4A2 P43354 2/20 0.70
GAA P10253 2/20 0.61
MAPT P10636 1/20 0.61
ATM Q13315 1/20 0.61
FADS1 O60427 1/20 0.59
PKM P14618 1/20 0.56
CYP1A2 P05177 9/20 0.55
CYP2D6 P10635 9/20 0.55
HPSE Q9Y251 2/20 0.54
CYP2C8 P10632 6/20 0.54
CYP2C19 P33261 6/20 0.54
KCNH2 Q12809 5/20 0.54
CYP2C9 P11712 4/20 0.54
CYP3A4 P08684 3/20 0.54
ABCB11 O95342 1/20 0.54
CHRM2 P08172 1/20 0.54
HTR1A P08908 1/20 0.54
CHRM1 P11229 1/20 0.54
DRD2 P14416 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Metaquine SCHEMBL7205743 0.87 FADS1 (0.71) APPNR4A2GAAMAPTATM
SCHEMBL30179800 0.83 GAA (0.73) APPNR4A2GAAMAPTATM
SCHEMBL2011565 0.83 GAA (0.73) APPNR4A2GAAMAPTATM
SCHEMBL29205238 0.82 APP (1.00) APPNR4A2GAAMAPTATM
SCHEMBL5309628 0.81 MAPT (0.74) APPNR4A2GAAMAPTATM
SCHEMBL19633680 0.81 FADS1 (0.63) APPNR4A2GAAMAPTATM
SCHEMBL16407130 0.80 APP (0.60) APPNR4A2GAAMAPTATM
SCHEMBL21346925 0.79 CYP1A2 (0.66) APPNR4A2GAAMAPTATM
SCHEMBL6995625 0.78 EGFR (0.69) APPNR4A2GAK
SCHEMBL4751350 0.78 CYP2D6 (0.58) APPNR4A2GAAMAPTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008135886-A2 QUINOLINE DERIVATIVES FOR USE IN THE INHIBITION OF THE GROWTH OF TUMOUR CELLS UNIVERSITY OF PRETORIA (ZA) 2008-11-13 WO disclosed