SCHEMBL4751350

SCHEMBL4751350

CC(=O)c1cccc(Nc2ccnc3cc(Cl)ccc23)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 9/20 0.58
CYP1A2 P05177 8/20 0.58
GAA P10253 3/20 0.58
MAPT P10636 2/20 0.58
ATM Q13315 1/20 0.58
APP P05067 2/20 0.58
NR4A2 P43354 2/20 0.58
ERBB2 P04626 1/20 0.57
PTK6 Q13882 1/20 0.57
FADS1 O60427 1/20 0.56
DNMT1 P26358 1/20 0.54
DNMT3A Q9Y6K1 1/20 0.54
GAK O14976 1/20 0.53
NPC1 O15118 1/20 0.52
CYP2C8 P10632 6/20 0.52
CYP2C19 P33261 6/20 0.52
KCNH2 Q12809 5/20 0.52
CYP2C9 P11712 4/20 0.52
CYP3A4 P08684 3/20 0.52
ABCB11 O95342 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21346925 0.89 CYP1A2 (0.66) CYP2D6CYP1A2GAAMAPTATM
SCHEMBL4751730 0.86 MAPT (0.70) CYP2D6CYP1A2GAAMAPTATM
Metaquine SCHEMBL7205743 0.85 FADS1 (0.71) CYP2D6CYP1A2GAAMAPTATM
SCHEMBL29200469 0.83 GAK (0.55) ERBB2PTK6DNMT1DNMT3AGAK
SCHEMBL14024396 0.82 CYP2D6 (0.52) CYP2D6CYP1A2GAAMAPTATM
SCHEMBL4748788 0.82 CYP2D6 (0.52) CYP2D6CYP1A2GAAMAPTATM
SCHEMBL2011565 0.81 GAA (0.73) CYP2D6CYP1A2GAAMAPTATM
SCHEMBL30179800 0.81 GAA (0.73) CYP2D6CYP1A2GAAMAPTATM
SCHEMBL2011014 0.80 CYP1A2 (0.67) CYP2D6CYP1A2GAAMAPTATM
SCHEMBL2015985 0.80 GAK (0.63) CYP2D6CYP1A2GAAMAPTATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008135886-A2 QUINOLINE DERIVATIVES FOR USE IN THE INHIBITION OF THE GROWTH OF TUMOUR CELLS UNIVERSITY OF PRETORIA (ZA) 2008-11-13 WO disclosed