SCHEMBL4751945

SCHEMBL4751945

CCOC(=O)c1c(-c2ccccc2)[nH]c(=O)n1C1CCCCC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 9/20 0.53
DRD2 P14416 8/20 0.53
DRD3 P35462 7/20 0.53
ALDH1A1 P00352 6/20 0.47
TSHR P16473 1/20 0.47
MAPK1 P28482 1/20 0.46
OPRM1 P35372 1/20 0.45
OPRD1 P41143 1/20 0.45
OPRK1 P41145 1/20 0.45
OGFRL1 Q5TC84 1/20 0.45
POLB P06746 1/20 0.45
HTT P42858 1/20 0.45
CASP3 P42574 1/20 0.45
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
CHRM2 P08172 1/20 0.43
CHRM4 P08173 1/20 0.43
CHRM5 P08912 1/20 0.43
CHRM1 P11229 1/20 0.43
CHRM3 P20309 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL885809 0.83 OPRM1 (0.47) DRD4DRD2DRD3ALDH1A1TSHR
SCHEMBL7169413 0.73 TDP1 (0.60) ALDH1A1TSHRMAPK1POLBGAA
SCHEMBL9894423 0.73 MAPT (0.54) ALDH1A1TSHRMAPK1OPRM1OPRD1
SCHEMBL25360981 0.71 ALDH1A1 (0.45) ALDH1A1TSHRMAPK1OPRM1OPRD1
SCHEMBL4281769 0.70 OGFRL1 (0.53) ALDH1A1TSHROPRM1OPRD1OPRK1
SCHEMBL4284918 0.70 OGFRL1 (0.53) ALDH1A1TSHROPRM1OPRD1OPRK1
SCHEMBL1260403 0.70 ALDH1A1 (0.49) ALDH1A1MAPK1OPRM1OPRD1OPRK1
SCHEMBL885834 0.69 MEN1 (0.46) DRD4DRD2DRD3ALDH1A1MAPK1
SCHEMBL9642259 0.69 DRD2 (0.64) DRD4DRD2DRD3ALDH1A1MAPK1
SCHEMBL8689759 0.68 SMN1; SMN2 (0.41) MAPK1HTTGAACHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008139941-A1 SUBSTITUTED IMIDAZOLE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-11-20 WO disclosed