SCHEMBL4752371

SCHEMBL4752371

CN1CCc2cc(NC(=O)C3(C)CCN3)ccc2C1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CLK2 P49760 1/20 0.42
CLK3 P49761 1/20 0.42
DYRK1A Q13627 1/20 0.42
ROCK2 O75116 6/20 0.40
TMPRSS2 O15393 1/20 0.39
RAB9A P51151 4/20 0.38
NPC1 O15118 3/20 0.38
DRD2 P14416 1/20 0.38
DRD3 P35462 1/20 0.38
CYP3A4 P08684 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3440779 0.81 CLK2 (0.42) CLK2CLK3DYRK1AROCK2TMPRSS2
SCHEMBL8127319 0.78 CLK2 (0.45) CLK2CLK3DYRK1AROCK2TMPRSS2
SCHEMBL3652815 0.78 NPC1 (0.49) CLK2CLK3DYRK1ATMPRSS2RAB9A
SCHEMBL20119168 0.77 TMPRSS2 (0.50) CLK2CLK3DYRK1AROCK2TMPRSS2
SCHEMBL8132355 0.75 PSMB8 (0.46) CLK2CLK3DYRK1AROCK2RAB9A
SCHEMBL20119296 0.74 KCNA1 (0.49) ROCK2RAB9ANPC1DRD2DRD3
SCHEMBL4751055 0.74 ALDH1A1 (0.45) ROCK2TMPRSS2RAB9ANPC1CYP3A4
SCHEMBL13012381 0.74 HPGD (0.44) RAB9ANPC1DRD2DRD3CYP3A4
SCHEMBL2248318 0.74 ACLY (0.53) ROCK2RAB9ANPC1CYP3A4ALDH1A1
SCHEMBL13347344 0.74 ALDH1A1 (0.50) TMPRSS2RAB9ANPC1CYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008135525-A2 SUBSTITUTED AZETIDINES, MANUFACTURING AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-11-13 WO disclosed
WO-2008135525-A2 SUBSTITUTED AZETIDINES, MANUFACTURING AND USE THEREOF AS MEDICAMENTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-11-13 WO disclosed