SCHEMBL4752572

SCHEMBL4752572

C[C@@H](OC(=O)N1CCN(C(=O)O[C@H](C)n2c(=O)[nH]c3ccccc32)CC1)n1c(=O)[nH]c2ccccc21

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.56
CHRM2 P08172 1/20 0.45
CHRM4 P08173 1/20 0.45
CHRM5 P08912 1/20 0.45
CHRM1 P11229 1/20 0.45
CHRM3 P20309 1/20 0.45
DAO P14920 1/20 0.42
PLD1 Q13393 3/20 0.41
PLD2 O14939 2/20 0.40
HSD11B1 P28845 1/20 0.40
P2RX7 Q99572 1/20 0.40
OPRM1 P35372 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4752476 0.76 SLC6A2 (0.40) ALDH1A1HPGD
SCHEMBL30838374 0.73 POLB (1.00) POLBDAOALDH1A1HPGDMEN1
SCHEMBL828232 0.73 POLB (1.00) POLBDAOALDH1A1HPGDMEN1
SCHEMBL4753544 0.71 CHRM2 (0.37) POLBCHRM2CHRM4CHRM1CHRM3
SCHEMBL904825 0.70 POLB (0.74) POLBDAOOPRM1ALDH1A1HPGD
SCHEMBL7017890 0.70 POLB (0.74) POLBDAOOPRM1ALDH1A1HPGD
SCHEMBL10736441 0.70 POLB (0.74) POLBDAOOPRM1ALDH1A1HPGD
SCHEMBL23997201 0.70 POLB (0.68) POLBDAOALDH1A1HPGDMEN1
SCHEMBL30336952 0.70 POLB (0.68) POLBDAOALDH1A1HPGDMEN1
SCHEMBL7513143 0.70 POLB (0.68) POLBDAOPLD1OPRM1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008139941-A1 SUBSTITUTED IMIDAZOLE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-11-20 WO disclosed