SCHEMBL4752824

SCHEMBL4752824

CC(=O)N(C)N1C[C@H](C(=O)c2ncccn2)C(c2cccc(F)c2C)[C@H](C(=O)c2ncccn2)C1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.34
CYP2D6 P10635 1/20 0.34
ABL1 P00519 2/20 0.34
LRRK2 Q5S007 2/20 0.34
OXTR P30559 1/20 0.33
HCRTR1 O43613 9/20 0.33
HCRTR2 O43614 9/20 0.33
PROKR1 Q8TCW9 1/20 0.32
RIPK1 Q13546 4/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4752708 0.84 MEN1 (0.43) TAAR1CYP2D6HCRTR1HCRTR2RIPK1
SCHEMBL4749426 0.82 EED (0.42) TAAR1CYP2D6RIPK1
SCHEMBL4749424 0.82 EED (0.42) TAAR1CYP2D6RIPK1
SCHEMBL4749432 0.79 CYP2D6 (0.34) TAAR1CYP2D6HCRTR1HCRTR2
SCHEMBL4749407 0.74 EED (0.32) RIPK1
SCHEMBL4023587 0.72 EED (0.41)
SCHEMBL4023583 0.72 EED (0.41)
SCHEMBL4026176 0.70 KMT2A (0.39) TAAR1CYP2D6HCRTR1HCRTR2
SCHEMBL4019575 0.69 EED (0.37) TAAR1CYP2D6PROKR1
SCHEMBL4019577 0.69 EED (0.37) TAAR1CYP2D6PROKR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008140810-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INCORPORATED (US) 2008-11-20 WO disclosed