SCHEMBL4752708

SCHEMBL4752708

Cc1c(F)cccc1C1[C@@H](C(=O)c2ncccn2)CN(C)C[C@H]1C(=O)c1ncccn1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
TAAR1 Q96RJ0 2/20 0.40
CYP2D6 P10635 1/20 0.40
MAPK1 P28482 1/20 0.40
HCRTR1 O43613 4/20 0.36
HCRTR2 O43614 4/20 0.36
RIPK1 Q13546 2/20 0.34
HRH4 Q9H3N8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4749432 0.87 CYP2D6 (0.34) MEN1KMT2ATAAR1CYP2D6HCRTR1
SCHEMBL4026176 0.84 KMT2A (0.39) MEN1KMT2ATAAR1CYP2D6MAPK1
SCHEMBL4752824 0.84 TAAR1 (0.34) TAAR1CYP2D6HCRTR1HCRTR2RIPK1
SCHEMBL4749426 0.83 EED (0.42) TAAR1CYP2D6RIPK1
SCHEMBL4749424 0.83 EED (0.42) TAAR1CYP2D6RIPK1
SCHEMBL4749201 0.82 MEN1 (0.44) MEN1KMT2ATAAR1CYP2D6MAPK1
SCHEMBL4748993 0.82 MEN1 (0.44) MEN1KMT2ATAAR1CYP2D6MAPK1
SCHEMBL4749407 0.75 EED (0.32) MEN1KMT2ARIPK1
SCHEMBL4752869 0.74 MEN1 (0.40) MEN1KMT2AMAPK1
SCHEMBL4751351 0.74 MEN1 (0.40) MEN1KMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008140810-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INCORPORATED (US) 2008-11-20 WO claimed
WO-2008140810-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INCORPORATED (US) 2008-11-20 WO disclosed