SCHEMBL4753869

SCHEMBL4753869

NC(C=O)N1CCN(C(=O)c2cc(C(F)(F)F)ccc2Cl)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.49
MAPK8 P45983 1/20 0.44
MAPK10 P53779 1/20 0.44
TSHR P16473 2/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
ALOX15 P16050 1/20 0.42
RORC P51449 2/20 0.42
RAB9A P51151 1/20 0.40
NR1I2 O75469 1/20 0.40
CACNA1B Q00975 1/20 0.40
KDM4E B2RXH2 1/20 0.40
CNR2 P34972 1/20 0.39
ALDH1A1 P00352 2/20 0.39
SLC6A9 P48067 1/20 0.39
ALOX5AP P20292 3/20 0.39
FEN1 P39748 3/20 0.39
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
TYK2 P29597 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4755194 0.84 TSHR (0.60) MAPK8MAPK10TSHRLMNATP53
Hydrochloric Acid SCHEMBL3466281 0.83 SCN5A (0.51) MAPK8MAPK10TSHRLMNATP53
Hydrochloric Acid SCHEMBL4753480 0.83 TSHR (0.59) MAPK8MAPK10TSHRLMNATP53
SCHEMBL3764364 0.79 KMT2A (0.56) KMT2AMAPK8MAPK10TSHRLMNA
SCHEMBL1222370 0.78 KMT2A (0.55) KMT2AMAPK8MAPK10TSHRLMNA
SCHEMBL4753812 0.77 P2RX7 (0.51) KMT2ATSHRLMNATP53ALOX15
SCHEMBL4753470 0.76 SCD (0.51) TSHR
SCHEMBL4753765 0.75 HCRTR1 (0.44) KDM4ESCN5ASCN9A
Hydrochloric Acid SCHEMBL3466569 0.75 SCD (0.50) TSHR
Hydrochloric Acid SCHEMBL3466376 0.74 HCRTR1 (0.43) KDM4ESCN5ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008157844-A1 NOVEL PIPERAZINE DERIVATIVES AS INHIBITORS OF STEAROYL-COA DESATURASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2008-12-24 WO disclosed