SCHEMBL4754043

SCHEMBL4754043

CNCCC(OCCNC(=O)OC)c1cccc(Cl)c1.COC(=O)NCCOC(CCN(C)C(=O)OC(C)(C)C)c1cccc(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.40
REN P00797 8/20 0.40
CYP3A4 P08684 3/20 0.40
NOS2 P35228 2/20 0.37
AOC3 Q16853 1/20 0.34
KDM4E B2RXH2 1/20 0.34
S1PR3 Q99500 1/20 0.34
GPR88 Q9GZN0 1/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
MAPT P10636 1/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP2C19 P33261 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
IDO1 P14902 1/20 0.34
AURKA O14965 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL499264 0.96 REN (0.39) RENCYP3A4AOC3KDM4ES1PR3
SCHEMBL498921 0.96 REN (0.39) RENCYP3A4AOC3KDM4ES1PR3
SCHEMBL498922 0.86 SLC6A4 (0.52) SLC6A4RENCYP3A4NOS2MEN1
SCHEMBL499203 0.86 SLC6A4 (0.52) SLC6A4RENCYP3A4NOS2MEN1
SCHEMBL4756782 0.85 IDO1 (0.37) RENNOS2KDM4EMEN1MAPT
SCHEMBL499224 0.81 AOC3 (0.40) AOC3KDM4EGPR88IDO1AURKA
SCHEMBL499588 0.80 IDO1 (0.39) RENKDM4EMEN1MAPTHTT
SCHEMBL499136 0.80 REN (0.49) RENCYP3A4
SCHEMBL499685 0.80 REN (0.49) RENCYP3A4
SCHEMBL4754002 0.77 SLC6A4 (0.56) SLC6A4CYP3A4NOS2CYP1A2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156816-A2 RENIN INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2008-12-24 WO disclosed