SCHEMBL4755529

SCHEMBL4755529

CNc1nc([C@H]2CC[C@@H](C(F)(F)F)CC2)n(-c2ccc(Cl)cc2)c(=O)c1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 4/20 0.39
DRD5 P21918 4/20 0.39
GRM1 Q13255 1/20 0.36
POLB P06746 2/20 0.36
KMT2A Q03164 1/20 0.36
AVPR1A P37288 2/20 0.35
MAT2A P31153 2/20 0.33
JUN P05412 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
KCNH2 Q12809 1/20 0.32
CRHR1 P34998 1/20 0.32
BRD4 O60885 1/20 0.32
BRD2 P25440 1/20 0.32
BRD3 Q15059 1/20 0.32
CREBBP Q92793 1/20 0.32
CNR1 P21554 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GSR P00390 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4755531 1.00 DRD1 (0.39) DRD1DRD5GRM1POLBKMT2A
SCHEMBL4756551 0.91 DRD1 (0.40) DRD1DRD5GRM1POLBKMT2A
SCHEMBL4755225 0.91 DRD1 (0.40) DRD1DRD5GRM1POLBKMT2A
SCHEMBL4755228 0.91 DRD1 (0.40) DRD1DRD5GRM1POLBKMT2A
SCHEMBL4755752 0.87 DRD1 (0.41) DRD1DRD5GRM1POLBKMT2A
SCHEMBL4755753 0.87 DRD1 (0.41) DRD1DRD5GRM1POLBKMT2A
SCHEMBL13985228 0.87 CRHR1 (0.35) DRD1DRD5AVPR1ACRHR1
SCHEMBL4911234 0.83 DRD1 (0.42) DRD1DRD5GRM1POLBKMT2A
SCHEMBL13985425 0.81 DRD1 (0.41) DRD1DRD5GRM1POLBKMT2A
SCHEMBL13985295 0.81 DRD1 (0.41) DRD1DRD5GRM1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008156607-A1 SUBSTITUTED PYRIMIDINONES NEUROGEN CORPORATION (US) 2008-12-24 WO claimed
WO-2008156607-A1 SUBSTITUTED PYRIMIDINONES NEUROGEN CORPORATION (US) 2008-12-24 WO disclosed
WO-2008156607-A1 SUBSTITUTED PYRIMIDINONES NEUROGEN CORPORATION (US) 2008-12-24 WO disclosed