SCHEMBL4756204

SCHEMBL4756204

CS(=O)(=O)Oc1cc(Cl)cc(C(=O)Nc2nccs2)c1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.52
BRD4 O60885 1/20 0.52
MAPT P10636 1/20 0.52
GCK P35557 9/20 0.52
RAB9A P51151 5/20 0.51
NPC1 O15118 3/20 0.51
HPGD P15428 1/20 0.51
HSD17B10 Q99714 1/20 0.49
KCNMA1 Q12791 1/20 0.48
MAPK1 P28482 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4755922 0.82 RAB9A (0.71) SMN1; SMN2RAB9ANPC1HPGDHSD17B10
SCHEMBL8797071 0.82 NPC1 (0.62) SMN1; SMN2BRD4MAPTGCKRAB9A
SCHEMBL706414 0.82 RAB9A (0.71) SMN1; SMN2MAPTGCKRAB9ANPC1
SCHEMBL6918311 0.76 GRM5 (0.53) SMN1; SMN2GCKRAB9ANPC1HPGD
SCHEMBL9070875 0.74 GCK (0.56) SMN1; SMN2BRD4MAPTGCKRAB9A
SCHEMBL2664747 0.74 RAB9A (0.77) SMN1; SMN2BRD4MAPTGCKRAB9A
SCHEMBL4756199 0.74 RAB9A (0.62) SMN1; SMN2BRD4MAPTRAB9ANPC1
SCHEMBL28801036 0.71 NPC1 (0.72) SMN1; SMN2MAPTGCKRAB9ANPC1
SCHEMBL14018616 0.71 RAB9A (0.72) SMN1; SMN2BRD4MAPTRAB9ANPC1
SCHEMBL2664728 0.71 GCK (0.60) SMN1; SMN2BRD4MAPTGCKRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8895752-B2 Alkylsulfonyl-substituted thiazolide compounds ROMARK LABORATORIES L.C. (US) 2014-11-25 US disclosed
US-8895752-B2 Alkylsulfonyl-substituted thiazolide compounds ROMARK LABORATORIES L.C. (US) 2014-11-25 US disclosed
US-20120122939-A1 ALKYLSULFONYL-SUBSTITUTED THIAZOLIDE COMPOUNDS ROMARK LABORATORIES, L.C. 2012-05-17 US disclosed
US-20120122939-A1 ALKYLSULFONYL-SUBSTITUTED THIAZOLIDE COMPOUNDS ROMARK LABORATORIES, L.C. 2012-05-17 US disclosed
US-8124632-B2 Alkylsulfonyl-substituted thiazolide compounds ROMARK LABORATORIES, L.C. (US) 2012-02-28 US disclosed
WO-2009035788-A1 ALKYLSULFONYL-SUBSTITUTED THIAZOLIDE COMPOUNDS ROMARK LABORATORIES L.C. (US) 2009-03-19 WO disclosed
US-20090036467-A1 ALKYLSULFONYL-SUBSTITUTED THIAZOLIDE COMPOUNDS ROMARK LABORATORIES L.C. 2009-02-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120122939-A1 ALKYLSULFONYL-SUBSTITUTED THIAZOLIDE COMPOUNDS HAVCR2, EIF2AK2, AADAC SMN1; SMN2 3410/4885BRD4 54/4885MAPT 4288/4885
US-20090036467-A1 ALKYLSULFONYL-SUBSTITUTED THIAZOLIDE COMPOUNDS HAVCR2, EIF2AK2, AADAC SMN1; SMN2 3410/4885BRD4 54/4885MAPT 4288/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.