SCHEMBL4757920

SCHEMBL4757920

COC(C(=O)O)c1nnc(-c2cc(Cl)cc(Cl)c2)o1.[NaH]

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 1/20 0.41
HPGD P15428 1/20 0.37
CTSA P10619 9/20 0.37
NOTUM Q6P988 1/20 0.36
TTR P02766 1/20 0.36
ALB P02768 1/20 0.36
MAOA P21397 1/20 0.36
CNR1 P21554 1/20 0.36
DRD1 P21728 1/20 0.36
OPRD1 P41143 1/20 0.36
PDE4D Q08499 1/20 0.36
PDE3A Q14432 1/20 0.36
TP53 P04637 2/20 0.34
NPC1 O15118 1/20 0.34
TSHR P16473 1/20 0.34
NFKB1 P19838 1/20 0.34
RAB9A P51151 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4757721 0.99 S1PR3 (0.42) S1PR3HPGDCTSANOTUMTTR
SCHEMBL4757922 0.85 S1PR3 (0.38) S1PR3HPGDCTSANOTUMTTR
SCHEMBL13985250 0.83 HSD17B10 (0.41) S1PR3CTSANPC1TSHRRAB9A
SCHEMBL9031273 0.71 NPC1 (0.44) S1PR3HPGDNOTUMTP53NPC1
SCHEMBL11125232 0.69 ALDH1A1 (0.40) SMN1; SMN2
SCHEMBL8626679 0.68
SCHEMBL4758257 0.65 RXRA (0.43) NOTUMTTRALBMAOACNR1
SCHEMBL2388785 0.65 TP53 (0.44) HPGDCTSATP53NPC1NFKB1
SCHEMBL10334912 0.65 KCNA5 (0.46) CTSACNR1
SCHEMBL1544916 0.63 NOTUM (0.52) NOTUMTP53NPC1TSHRNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000819-A1 5-PHENYL-1,3,4-OXADIAZOL-2-YL-ACETYL-4-PIPERIDINYL DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2008-12-31 WO disclosed