SCHEMBL8626679

SCHEMBL8626679

COC(C(=O)O)c1nnc(S)o1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4757721 0.69 S1PR3 (0.42)
SCHEMBL4757920 0.68 S1PR3 (0.41)
SCHEMBL8628308 0.68
SCHEMBL24328842 0.64 CTSA (0.40)
SCHEMBL8628463 0.64
SCHEMBL24327736 0.64 CTSA (0.40)
SCHEMBL8627742 0.64 GLS (0.31)
SCHEMBL3827990 0.64 C3AR1 (0.34)
SCHEMBL23424110 0.59 NR4A2 (0.37)
SCHEMBL24328853 0.58 IMPDH2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE35754-E FOR TREATING BACTERIAL INFECTIONS HOECHST AKTIENGESELLSCHAFT (DE) 1998-03-24 US disclosed
US-5710146-A ANTIBIOTICS FOR BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1998-01-20 US disclosed
US-5089490-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1992-02-18 US disclosed
US-4758556-A Cephem derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1988-07-19 US disclosed
US-4278793-A ANTIBIOTICS, BACTERICIDES HOECHST AKTIENGESELLSCHAFT (DE) 1981-07-14 US disclosed
US-4183925-A 7-Aminophenylacetamido-Δ3 -cephem antibacterial agents and method of use PFIZER INC. (US) 1980-01-15 US disclosed
US-4144240-A USED FOR MODIFYING CEPHALOSPORINS PFIZER INC. (US) 1979-03-13 US disclosed