SCHEMBL4759150

SCHEMBL4759150

CC(C)(Sc1ccc(Cl)cc1)C(=O)N1CCC2(C1)OCc1ccccc12

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 15/20 0.46
OXTR P30559 1/20 0.46
HRH3 Q9Y5N1 1/20 0.42
AVPR2 P30518 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4759147 1.00 AVPR1A (0.46) AVPR1AOXTRHRH3AVPR2
SCHEMBL4759117 0.82 HSD11B1 (0.61) AVPR1AHRH3
SCHEMBL4759115 0.82 HSD11B1 (0.61) AVPR1AHRH3
SCHEMBL3682438 0.80 AVPR1A (0.48) AVPR1AOXTRHRH3AVPR2
SCHEMBL349521 0.76 HSD11B1 (0.67) AVPR1AOXTR
SCHEMBL18701840 0.74 AVPR1A (0.58) AVPR1AOXTRHRH3AVPR2
SCHEMBL3232343 0.74 AVPR1A (0.57) AVPR1AHRH3AVPR2
SCHEMBL3231283 0.74 AVPR1A (0.54) AVPR1AOXTRHRH3AVPR2
SCHEMBL5531225 0.73 AVPR1A (0.53) AVPR1AOXTRHRH3AVPR2
SCHEMBL4757502 0.73 HSD11B1 (0.52) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1758582-A4 AMIDO COMPOUNDS AND THEIR USE AS PHARMACEUTICALS INCYTE CORP (US) 2008-01-09 EP claimed
EP-1758582-A1 AMIDO COMPOUNDS AND THEIR USE AS PHARMACEUTICALS Incyte Corporation (US) 2007-03-07 EP claimed
US-20060009471-A1 Amido compounds and their use as pharmaceuticals INCYTE CORPORATION 2006-01-12 US claimed
WO-2006002349-A1 AMIDO COMPOUNDS AND THEIR USE AS PHARMACEUTICALS INCYTE CORPORATION (US) 2006-01-05 WO claimed
EP-1758582-A4 AMIDO COMPOUNDS AND THEIR USE AS PHARMACEUTICALS INCYTE CORP (US) 2008-01-09 EP disclosed
EP-1758582-A1 AMIDO COMPOUNDS AND THEIR USE AS PHARMACEUTICALS Incyte Corporation (US) 2007-03-07 EP disclosed
US-20060009471-A1 Amido compounds and their use as pharmaceuticals INCYTE CORPORATION 2006-01-12 US disclosed
WO-2006002349-A1 AMIDO COMPOUNDS AND THEIR USE AS PHARMACEUTICALS INCYTE CORPORATION (US) 2006-01-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060009471-A1 Amido compounds and their use as pharmaceuticals HSD11B1, CYP11B1, HSD11B2 AVPR1A 60/4885OXTR 367/4885HRH3 1465/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.