SCHEMBL4759738

SCHEMBL4759738

COc1cc(C(=O)[C@H]2C(=O)c3cc(N4CCNCC4)ccc3OC23CCNCC3)nc2c(OC)cccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 2/20 0.38
ACACB O00763 1/20 0.38
ACACA Q13085 1/20 0.38
DCLK1 O15075 1/20 0.36
MAPK7 Q13164 1/20 0.36
LRRK2 Q5S007 1/20 0.36
HTR1A P08908 1/20 0.36
PDE7A Q13946 3/20 0.35
ALK Q9UM73 7/20 0.34
PDE4D Q08499 1/20 0.34
PDE7B Q9NP56 1/20 0.34
TNF P01375 1/20 0.34
LITAF Q99732 1/20 0.34
CDK2 P24941 1/20 0.33
CDK9 P50750 1/20 0.33
CDK5 Q00535 1/20 0.33
ABCB1 P08183 1/20 0.33
ADRB1 P08588 1/20 0.33
TGFBR1 P36897 1/20 0.33
ACVR1 Q04771 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4760231 0.93 ALK (0.40) ACACBACACAPDE7AALK
SCHEMBL4708583 0.87 XIAP (0.39) ACACBACACA
SCHEMBL4707073 0.87 ACACB (0.35) ACACBACACATNFLITAF
SCHEMBL4707267 0.87 ACACA (0.38) ACACBACACA
SCHEMBL4708596 0.87 ACACA (0.36) ACACBACACATNFLITAF
SCHEMBL4708996 0.85 ACACA (0.35) ACACBACACATNFLITAF
SCHEMBL4710103 0.84 ACACA (0.37) ACACBACACATNFLITAF
SCHEMBL4760480 0.84 NOTUM (0.36) ACACBACACAPDE7A
SCHEMBL4759663 0.84 TTK (0.37) ACACBACACA
SCHEMBL4709980 0.83 ACACA (0.36) ACACBACACACDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910375-A1 SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS Merck & Co., Inc. (US) 2008-04-16 EP disclosed
WO-2007011809-A1 SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS MERCK & CO., INC. (US) 2007-01-25 WO disclosed