SCHEMBL4709980

SCHEMBL4709980

COc1cc(C(=O)[C@H]2C(=O)c3c[c]ccc3OC23CCNCC3)nc2c(OC)cccc12

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACACA Q13085 2/20 0.36
ACACB O00763 1/20 0.36
JUND P17535 1/20 0.33
FOSB P53539 1/20 0.33
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
HPGD P15428 2/20 0.31
CDK2 P24941 1/20 0.30
XIAP P98170 1/20 0.30
PDE10A Q9Y233 1/20 0.30
HSD17B10 Q99714 1/20 0.30
TNKS O95271 1/20 0.30
PARP1 P09874 1/20 0.30
TNKS2 Q9H2K2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4707267 0.89 ACACA (0.38) ACACAACACBJUNDFOSBKDM4E
SCHEMBL4708583 0.86 XIAP (0.39) ACACAACACBJUNDFOSBKDM4E
SCHEMBL4708596 0.85 ACACA (0.36) ACACAACACBJUNDFOSBKDM4E
SCHEMBL4708996 0.83 ACACA (0.35) ACACAACACBJUNDFOSBKDM4E
SCHEMBL4759738 0.83 HTR7 (0.38) ACACAACACBCDK2
SCHEMBL4710103 0.83 ACACA (0.37) ACACAACACBJUNDFOSBPDE10A
SCHEMBL4759789 0.82 TNKS (0.34) ACACAACACBJUNDFOSBXIAP
SCHEMBL4760214 0.82 ACACA (0.34) ACACAACACBJUNDFOSBTNKS
SCHEMBL4760480 0.81 NOTUM (0.36) ACACAACACBKDM4EALDH1A1HSD17B10
SCHEMBL2362040 0.81 ACACB (0.35) ACACAACACBJUNDFOSBTNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910375-A1 SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS Merck & Co., Inc. (US) 2008-04-16 EP disclosed
WO-2007011811-A1 SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS MERCK & CO., INC. (US) 2007-01-25 WO disclosed
WO-2007011809-A1 SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS MERCK & CO., INC. (US) 2007-01-25 WO disclosed