SCHEMBL4708596

SCHEMBL4708596

COc1cc(C(=O)[C@H]2C(=O)c3cc(C(=O)O)ccc3OC23CCNCC3)nc2c(OC)cccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACA Q13085 2/20 0.36
ACACB O00763 2/20 0.36
PDE10A Q9Y233 1/20 0.34
ALOX15 P16050 1/20 0.33
SSTR5 P35346 1/20 0.33
JUND P17535 1/20 0.33
FOSB P53539 1/20 0.33
OPRD1 P41143 2/20 0.32
XIAP P98170 2/20 0.32
GPR35 Q9HC97 1/20 0.31
TNKS O95271 1/20 0.31
TNKS2 Q9H2K2 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
HPGD P15428 2/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
TNF P01375 1/20 0.30
LITAF Q99732 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708583 0.89 XIAP (0.39) ACACAACACBJUNDFOSBXIAP
SCHEMBL4707267 0.89 ACACA (0.38) ACACAACACBPDE10AALOX15JUND
SCHEMBL4707168 0.89 MEN1 (0.36) ACACAACACBKDM4EALDH1A1LMNA
SCHEMBL4708996 0.88 ACACA (0.35) ACACAACACBPDE10AJUNDFOSB
SCHEMBL4710103 0.88 ACACA (0.37) ACACAACACBPDE10AJUNDFOSB
SCHEMBL4759738 0.87 HTR7 (0.38) ACACAACACBTNFLITAF
SCHEMBL4760214 0.86 ACACA (0.34) ACACAACACBJUNDFOSBTNKS
SCHEMBL4710002 0.86 ACACB (0.36) ACACAACACBLMNATP53
SCHEMBL4709980 0.85 ACACA (0.36) ACACAACACBPDE10AJUNDFOSB
SCHEMBL4759789 0.85 TNKS (0.34) ACACAACACBJUNDFOSBXIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910375-A1 SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS Merck & Co., Inc. (US) 2008-04-16 EP claimed
WO-2007011809-A1 SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS MERCK & CO., INC. (US) 2007-01-25 WO claimed