SCHEMBL4760688

SCHEMBL4760688

Nc1nn2ccnc2c(N)c1-c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.41
RAB9A P51151 4/20 0.41
MAPT P10636 4/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
JAK2 O60674 7/20 0.40
JAK3 P52333 7/20 0.40
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
GAA P10253 2/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
ADORA2A P29274 1/20 0.37
EGFR P00533 1/20 0.36
SRC P12931 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
SYK P43405 1/20 0.36
CDK8 P49336 1/20 0.36
ACVR1 Q04771 1/20 0.36
AKT1 P31749 1/20 0.35
NUDT1 P36639 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4757863 0.87 NUDT1 (0.35) NPC1RAB9AMAPTSMN1; SMN2JAK2
SCHEMBL4709570 0.84 KDM4E (0.38) NPC1RAB9AMAPTSMN1; SMN2JAK2
SCHEMBL5453382 0.83 KDM4E (0.37) NPC1RAB9AMAPTSMN1; SMN2JAK2
SCHEMBL4759759 0.73 JAK2 (0.35) JAK2JAK3NUDT1
SCHEMBL13841918 0.70 KDM4E (0.49) NPC1RAB9AMAPTSMN1; SMN2MEN1
SCHEMBL5741027 0.70 SMPD3 (0.50) JAK2JAK3NUDT1
SCHEMBL13841874 0.69 PIK3CG (0.51) NPC1RAB9AMAPTSMN1; SMN2JAK2
SCHEMBL3703475 0.69 JAK2 (0.55) NPC1MAPTJAK2JAK3NPSR1
Hydrochloric Acid SCHEMBL3022279 0.68 NPC1 (0.36) NPC1RAB9AMAPTSMN1; SMN2KMT2A
SCHEMBL12145626 0.67 TSHR (0.47) MAPTMEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928879-A2 FUSED HETEROCYCLIC COMPOUNDS USEFUL AS KINASE MODULATORS Brystol-Myers Squibb Company (US) 2008-06-11 EP claimed
WO-2007038314-A2 FUSED HETEROCYCLIC COMPOUNDS USEFUL AS KINASE MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-04-05 WO claimed