SCHEMBL4709570

SCHEMBL4709570

Cc1ccc(-c2c(N)nn3ccnc3c2N)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.38
SRC P12931 3/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
FYN P06241 2/20 0.38
KDR P35968 2/20 0.38
PLK4 O00444 1/20 0.38
RIPK2 O43353 1/20 0.38
ROCK2 O75116 1/20 0.38
PRKD3 O94806 1/20 0.38
MAP4K4 O95819 1/20 0.38
ABL1 P00519 1/20 0.38
EGFR P00533 1/20 0.38
LMNA P02545 1/20 0.38
ERBB2 P04626 1/20 0.38
INSR P06213 1/20 0.38
LCK P06239 1/20 0.38
CSF1R P07333 1/20 0.38
YES1 P07947 1/20 0.38
LYN P07948 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5453382 0.98 KDM4E (0.37) KDM4ESRCALDH1A1HPGDFYN
SCHEMBL4757863 0.88 NUDT1 (0.35) KDM4EALDH1A1HPGDKDRKMT2A
SCHEMBL4760688 0.84 NPC1 (0.41) KDM4ESRCALDH1A1HPGDEGFR
SCHEMBL4759759 0.71 JAK2 (0.35) JAK2JAK3NUDT1
SCHEMBL3703475 0.67 JAK2 (0.55) NPSR1JAK2JAK3NPC1MAPT
SCHEMBL13841956 0.65 MAPT (0.52) KDM4EALDH1A1HPGDKDRPLK4
SCHEMBL19766651 0.65 NUDT1 (0.41) KDM4EALDH1A1HPGDLMNATSHR
SCHEMBL5741027 0.64 SMPD3 (0.50) MAP4K4JAK2JAK3NUDT1
SCHEMBL615165 0.63 ACHE (0.50) KDM4EALDH1A1HPGDLMNAMAPK1
SCHEMBL25333334 0.63 MAT2A (0.51) ALDH1A1MAPK14CYP1A2CYP3A4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928879-A2 FUSED HETEROCYCLIC COMPOUNDS USEFUL AS KINASE MODULATORS Brystol-Myers Squibb Company (US) 2008-06-11 EP claimed
WO-2007038314-A2 FUSED HETEROCYCLIC COMPOUNDS USEFUL AS KINASE MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-04-05 WO claimed