SCHEMBL4760729

SCHEMBL4760729

O=C(O)c1cn(C2CCCCC2)[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.43
HSD17B10 Q99714 5/20 0.36
ALDH1A1 P00352 3/20 0.36
KDM6B O15054 1/20 0.36
KDM4A O75164 1/20 0.36
KDM4D Q6B0I6 1/20 0.36
KDM3B Q7LBC6 1/20 0.36
HIF1AN Q9NWT6 1/20 0.36
KDM2A Q9Y2K7 1/20 0.36
GAA P10253 3/20 0.35
HPGD P15428 2/20 0.35
POLB P06746 1/20 0.35
ACMSD Q8TDX5 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
LDHA P00338 1/20 0.33
DDO Q99489 1/20 0.33
UCHL1 P09936 1/20 0.33
EPHX2 P34913 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL692076 0.68 ALDH1A1 (0.41) KDM4EHSD17B10ALDH1A1GAAPOLB
SCHEMBL10208596 0.64 KDM4E (0.48) KDM4EHSD17B10ALDH1A1GAAHPGD
SCHEMBL19377738 0.64 AXL (0.40) KDM4EHSD17B10ALDH1A1HIF1ANGAA
SCHEMBL30612395 0.62 KDM4E (0.52) KDM4EHSD17B10ALDH1A1GAAHPGD
SCHEMBL11054514 0.62 HCAR1 (0.38) KDM4EALDH1A1KMT2AEPHX2
SCHEMBL21785477 0.62 AXL (0.38) KDM4EHSD17B10ALDH1A1HIF1ANGAA
Hydrochloric Acid SCHEMBL11452778 0.61 KDM4E (0.51) KDM4EHSD17B10ALDH1A1GAAHPGD
SCHEMBL15486621 0.61 KDM4E (0.48) KDM4EHSD17B10ALDH1A1GAAHPGD
SCHEMBL925044 0.60 KDM4E (0.64) KDM4EHSD17B10ALDH1A1GAAHPGD
SCHEMBL924129 0.60 HSD17B10 (0.51) KDM4EHSD17B10ALDH1A1GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1999114-A2 PYRAZOLES AS 11-BETA-HSD-1 F. Hoffmann-la Roche AG (CH) 2008-12-10 EP disclosed
WO-2007107470-A2 PYRAZOLES AS 11-BETA-HSD-1 F. HOFFMANN-LA ROCHE AG (CH) 2007-09-27 WO disclosed