SCHEMBL4763441

SCHEMBL4763441

O=c1c([N+](=O)[O-])c(/C=C/c2cnn(Cc3ccccc3F)c2)n(CCc2ccccc2)c(=O)n1C1CCC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.34
TSHR P16473 2/20 0.34
NPSR1 Q6W5P4 3/20 0.33
ALDH1A1 P00352 3/20 0.33
POLB P06746 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
MAPT P10636 4/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PDE1A P54750 1/20 0.33
PDE1B Q01064 1/20 0.33
PDE1C Q14123 1/20 0.33
PKM P14618 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HDAC2 Q92769 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4766007 0.91 C5AR1 (0.41) ADORA2AADORA2BADORA1C5AR1
SCHEMBL4769541 0.88 MAPT (0.37) ALDH1A1ADORA2AADORA2BADORA1MAPT
SCHEMBL4765722 0.88 TP53 (0.41) TP53TSHRALDH1A1ADORA2AADORA2B
SCHEMBL4769532 0.88 MAPT (0.37) ALDH1A1ADORA2AADORA2BADORA1MAPT
SCHEMBL4765708 0.88 TP53 (0.41) TP53TSHRALDH1A1ADORA2AADORA2B
SCHEMBL4771507 0.86 MAPT (0.36) NPSR1ALDH1A1POLBMAPTSMN1; SMN2
SCHEMBL4867818 0.85 ADORA2B (0.39) TP53TSHRNPSR1ALDH1A1POLB
SCHEMBL4792629 0.84 SMN1; SMN2 (0.35) TSHRNPSR1ALDH1A1POLBMAPT
SCHEMBL4763924 0.84 NPSR1 (0.33) TSHRNPSR1ALDH1A1POLBADORA2A
SCHEMBL4763921 0.84 NPSR1 (0.33) TSHRNPSR1ALDH1A1POLBADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678181-B1 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS INC (US) 2008-12-31 EP disclosed