SCHEMBL4765722

SCHEMBL4765722

O=c1c([N+](=O)[O-])c(C=Cc2cnn(Cc3ccccc3F)c2)n(CCc2ccccc2)c(=O)n1CCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.41
ADORA2B P29275 2/20 0.40
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
MAPT P10636 3/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
ALDH1A1 P00352 2/20 0.37
PKM P14618 2/20 0.37
LMNA P02545 1/20 0.36
HDAC2 Q92769 2/20 0.36
GAA P10253 1/20 0.35
THRB P10828 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
TSHR P16473 1/20 0.34
HSPD1 P10809 1/20 0.34
HSPE1 P61604 1/20 0.34
PSD A5PKW4 1/20 0.33
PKLR P30613 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4765708 1.00 TP53 (0.41) TP53ADORA2BADORA2AADORA1MAPT
SCHEMBL4771531 0.93 ADORA2B (0.38) TP53ADORA2BADORA2AADORA1MAPT
SCHEMBL4771549 0.93 ADORA2B (0.38) TP53ADORA2BADORA2AADORA1MAPT
SCHEMBL4763171 0.90 ADORA2B (0.43) TP53ADORA2BADORA2AADORA1MAPT
SCHEMBL4763165 0.90 ADORA2B (0.43) TP53ADORA2BADORA2AADORA1MAPT
SCHEMBL4764053 0.89 ALDH1A1 (0.41) TP53ADORA2BADORA2AADORA1MAPT
SCHEMBL4763441 0.88 TP53 (0.34) TP53ADORA2BADORA2AADORA1MAPT
SCHEMBL4763896 0.88 ADORA2B (0.46) ADORA2BADORA2AADORA1MAPTL3MBTL1
SCHEMBL4763889 0.88 ADORA2B (0.46) ADORA2BADORA2AADORA1MAPTL3MBTL1
SCHEMBL4771427 0.87 ADORA2B (0.41) TP53ADORA2BADORA2AADORA1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678181-B1 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS INC (US) 2008-12-31 EP disclosed