SCHEMBL4764668

SCHEMBL4764668

O=C(N[C@@H](Cc1ccccc1)C(=O)O)c1ccc(Cn2ccc3cc(N(c4ccccc4)S(=O)(=O)c4ccccc4)ccc32)cc1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.49
CA12 O43570 2/20 0.49
CA9 Q16790 2/20 0.49
PTPN1 P18031 2/20 0.48
CA2 P00918 7/20 0.47
MEN1 O00255 2/20 0.45
ALDH1A1 P00352 2/20 0.45
KMT2A Q03164 2/20 0.45
ITGB1 P05556 1/20 0.43
ITGA4 P13612 1/20 0.43
PPARG P37231 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NTSR1 P30989 1/20 0.43
ACE P12821 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3193347 0.82 CA2 (0.49) CA1PTPN1CA2MEN1ALDH1A1
SCHEMBL3193462 0.78 SERPINE1 (0.53) CA1CA2MEN1ALDH1A1KMT2A
SCHEMBL3204698 0.76 NR1I2 (0.53) CA1CA12CA9CA2MEN1
SCHEMBL3185435 0.74 SERPINE1 (0.52) CA1CA2MEN1ALDH1A1KMT2A
SCHEMBL3202333 0.71 PPARG (0.49) PPARGNTSR1ACE
SCHEMBL3202345 0.71 PPARG (0.49) PPARGNTSR1ACE
SCHEMBL3186142 0.70 FPR2 (0.53)
SCHEMBL27718316 0.70 FPR2 (0.53)
SCHEMBL3195456 0.68 TRPM8 (0.51) MEN1ALDH1A1KMT2A
SCHEMBL3197128 0.68 PPARG (0.53) CA2PPARGSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919866-A2 SUBSTITUTED INDOLES AND USE THEREOF Wyeth a Corporation of the State of Delaware (US) 2008-05-14 EP claimed
WO-2007022321-A2 SUBSTITUTED INDOLES AND USE THEREOF WYETH (US) 2007-02-22 WO claimed