SCHEMBL476472

SCHEMBL476472

CC(F)(OC(N)=O)c1ccccn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
AHR P35869 1/20 0.41
CETP P11597 5/20 0.41
MAPK1 P28482 1/20 0.41
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
RAB9A P51151 1/20 0.40
BLM P54132 2/20 0.39
CYP2D6 P10635 1/20 0.39
SLC22A2 O15244 1/20 0.39
SLC22A1 O15245 1/20 0.39
PGR P06401 1/20 0.39
THRB P10828 1/20 0.39
ADRB3 P13945 1/20 0.39
OPRK1 P41145 1/20 0.39
PMP22 Q01453 1/20 0.39
KCNH2 Q12809 1/20 0.39
PDE3A Q14432 1/20 0.39
SLC47A1 Q96FL8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2465547 0.83 SMN1; SMN2 (0.46) SMN1; SMN2L3MBTL1AHRCETPMAPK1
SCHEMBL29137044 0.81 SMN1; SMN2 (0.43) SMN1; SMN2L3MBTL1AHRCETPMAPK1
SCHEMBL2465434 0.78 SMN1; SMN2 (0.50) SMN1; SMN2L3MBTL1AHRMAPK1NPC1
SCHEMBL30211312 0.77 AHR (0.40) SMN1; SMN2L3MBTL1AHRCETPMAPK1
SCHEMBL8283520 0.74 MAPT (0.52) SMN1; SMN2L3MBTL1MAPK1NPC1TP53
SCHEMBL20166133 0.73 AHR (0.47) SMN1; SMN2L3MBTL1AHRNPC1TP53
SCHEMBL21742399 0.73 SMN1; SMN2 (0.42) SMN1; SMN2L3MBTL1AHRCETPNPC1
SCHEMBL28996600 0.73 SMN1; SMN2 (0.48) SMN1; SMN2L3MBTL1MAPK1NPC1TP53
SCHEMBL1026708 0.73 L3MBTL1 (0.48) SMN1; SMN2L3MBTL1AHRCETPBLM
Acetic Acid SCHEMBL28062268 0.73 L3MBTL1 (0.48) SMN1; SMN2L3MBTL1AHRCETPBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2410858-A1 P2X3 RECEPTOR ANTAGONISTS FOR TREATMENT OF PAIN Merck Sharp & Dohme Corp. (US) 2012-02-01 EP disclosed
WO-2010111059-A1 P2X3 RECEPTOR ANTAGONISTS FOR TREATMENT OF PAIN MERCK SHARP & DOHME CORP. (US) 2010-09-30 WO disclosed