SCHEMBL29137044

SCHEMBL29137044

CC(C)(C)C(C)(OC(N)=O)c1ccccn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MAPK1 P28482 1/20 0.41
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
RAB9A P51151 1/20 0.40
BLM P54132 2/20 0.39
CYP2D6 P10635 1/20 0.39
SLC22A2 O15244 1/20 0.39
SLC22A1 O15245 1/20 0.39
PGR P06401 1/20 0.39
THRB P10828 1/20 0.39
ADRB3 P13945 1/20 0.39
OPRK1 P41145 1/20 0.39
PMP22 Q01453 1/20 0.39
KCNH2 Q12809 1/20 0.39
PDE3A Q14432 1/20 0.39
SLC47A1 Q96FL8 1/20 0.39
CYP3A4 P08684 1/20 0.39
ALOX15 P16050 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21742051 0.85 L3MBTL1 (0.44) SMN1; SMN2L3MBTL1MAPK1NPC1TP53
SCHEMBL2465547 0.83 SMN1; SMN2 (0.46) SMN1; SMN2L3MBTL1MAPK1NPC1TP53
SCHEMBL476472 0.81 SMN1; SMN2 (0.43) SMN1; SMN2L3MBTL1MAPK1NPC1TP53
SCHEMBL29188178 0.79 P2RX7 (0.36) KMT2A
SCHEMBL21742069 0.75 SMN1; SMN2 (0.47) SMN1; SMN2L3MBTL1NPC1RAB9ABLM
SCHEMBL8283520 0.74 MAPT (0.52) SMN1; SMN2L3MBTL1MAPK1NPC1TP53
SCHEMBL21742399 0.73 SMN1; SMN2 (0.42) SMN1; SMN2L3MBTL1NPC1RAB9ABLM
SCHEMBL28996600 0.73 SMN1; SMN2 (0.48) SMN1; SMN2L3MBTL1MAPK1NPC1TP53
SCHEMBL21742276 0.73 SMN1; SMN2 (0.44) SMN1; SMN2L3MBTL1BLMCYP2D6KCNH2
SCHEMBL27205053 0.72 SMN1; SMN2 (0.44) SMN1; SMN2L3MBTL1MAPK1NPC1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115551862-B Macrocyclic inhibitors of peptidyl arginine deiminase 吉利德科学公司 2024-04-12 CN disclosed
CN-117355521-A Heteroaryl inhibitors of plasma kallikrein 武田药品工业株式会社 2024-01-05 CN disclosed