SCHEMBL4764950

SCHEMBL4764950

CC(C)C[CH]C(=O)N(Cc1ccc2ccccc2n1)[C@H]1CCCNCC1=O

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
AGTR2 P50052 1/20 0.33
ALOX5AP P20292 1/20 0.33
ALOX5 P09917 7/20 0.33
HDAC6 Q9UBN7 1/20 0.33
REN P00797 1/20 0.32
HCRTR1 O43613 3/20 0.32
HCRTR2 O43614 3/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6590687 0.78 CXCR4 (0.32)
SCHEMBL4766714 0.75 GHSR (0.37) SLC6A2SLC6A4SLC6A3
SCHEMBL6608111 0.72 SLC6A2 (0.40) CYP2D6SLC6A2SLC6A4SLC6A3
SCHEMBL4761916 0.70 PSEN1 (0.33)
SCHEMBL6590845 0.70 ALDH1A1 (0.38) CYP3A4CYP2C19
SCHEMBL6590944 0.70 PSEN1 (0.31)
SCHEMBL4770129 0.69 LMNA (0.37) CYP1A2CYP3A4CYP2C19SLC6A2SLC6A3
SCHEMBL6591064 0.69
SCHEMBL6589898 0.69
SCHEMBL4762983 0.68 PSEN1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1320370-A4 METHOD OF TREATMENT SMITHKLINE BEECHAM CORP (US) 2008-10-22 EP disclosed
EP-1320370-A1 METHOD OF TREATMENT SmithKline Beecham Corporation (US) 2003-06-25 EP disclosed
WO-2002017924-A1 METHOD OF TREATMENT SMITHKLINE BEECHAM CORPORATION (GB) 2002-03-07 WO disclosed