SCHEMBL4765953

SCHEMBL4765953

O=C(CCc1nc(-c2ccccn2)no1)Nc1cc(-c2cccnc2)nc(-c2ccccn2)n1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.52
PKM P14618 5/20 0.51
HTT P42858 3/20 0.51
NPC1 O15118 3/20 0.51
RAB9A P51151 3/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
TP53 P04637 1/20 0.51
TSHR P16473 1/20 0.51
HDAC1 Q13547 2/20 0.50
HDAC2 Q92769 2/20 0.50
ALDH1A1 P00352 2/20 0.50
TDP1 Q9NUW8 1/20 0.49
KLF5 Q13887 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
MAPK1 P28482 3/20 0.48
CASP1 P29466 1/20 0.48
CYP2C9 P11712 1/20 0.48
HCAR2 Q8TDS4 1/20 0.48
USP2 O75604 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4775234 0.96 LMNA (0.49) LMNAPKMHTTNPC1RAB9A
SCHEMBL4766014 0.85 ADORA1 (0.47) LMNAPKMHTTNPC1RAB9A
SCHEMBL4768829 0.84 KDM4E (0.44) LMNAPKMNPC1RAB9ASMN1; SMN2
SCHEMBL4769061 0.84 ADORA2A (0.43) LMNAPKMHTTNPC1RAB9A
SCHEMBL4771450 0.82 NPC1 (0.52) LMNAPKMHTTNPC1RAB9A
SCHEMBL4775920 0.81 ADORA1 (0.54) LMNANPC1RAB9AHDAC1HDAC2
SCHEMBL4771758 0.81 ADORA1 (0.43) PKMHTTNPC1RAB9ASMN1; SMN2
SCHEMBL4773065 0.80 ADORA1 (0.43) PKMNPC1RAB9ASMN1; SMN2TP53
SCHEMBL4769102 0.80 KMT2A (0.55) LMNANPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL4770635 0.79 CYP1A2 (0.52) SMN1; SMN2TSHRALDH1A1TDP1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878733-A1 Pyrimidine derivatives as ALK-5 inhibitors Novartis AG (CH) 2008-01-16 EP disclosed