SCHEMBL4771758

SCHEMBL4771758

O=C(CCc1ncc[nH]1)Nc1cc(-c2cccnc2)nc(-c2ccccn2)n1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 8/20 0.43
ADORA2A P29274 7/20 0.43
ADORA3 P0DMS8 6/20 0.43
HTT P42858 1/20 0.41
CYP2A6 P11509 1/20 0.41
ADORA2B P29275 1/20 0.40
SCN5A Q14524 1/20 0.40
SCN9A Q15858 1/20 0.40
NPC1 O15118 2/20 0.39
TP53 P04637 2/20 0.39
PKM P14618 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KMT2A Q03164 1/20 0.39
TSHR P16473 1/20 0.39
GLA P06280 1/20 0.38
POLB P06746 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ATR Q13535 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4770635 0.86 CYP1A2 (0.52) ADORA1ADORA2AADORA3SMN1; SMN2TSHR
SCHEMBL4766014 0.85 ADORA1 (0.47) ADORA1ADORA2AADORA3HTTCYP2A6
SCHEMBL4773065 0.82 ADORA1 (0.43) ADORA1ADORA2AADORA3CYP2A6ADORA2B
SCHEMBL4773067 0.82 CYP3A4 (0.50) HTTCYP2A6NPC1TP53PKM
SCHEMBL4769102 0.82 KMT2A (0.55) ADORA1ADORA2AADORA3NPC1RAB9A
SCHEMBL4768684 0.82 ADORA2A (0.43) ADORA1ADORA2AADORA3CYP2A6ADORA2B
SCHEMBL4765953 0.81 LMNA (0.52) HTTNPC1TP53PKMRAB9A
SCHEMBL4775920 0.79 ADORA1 (0.54) ADORA1ADORA2AADORA3ADORA2BNPC1
SCHEMBL4768829 0.79 KDM4E (0.44) ADORA1ADORA2AADORA3CYP2A6ADORA2B
SCHEMBL4769062 0.79 ADRB2 (0.46) ADORA1ADORA2AADORA3HTTCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878733-A1 Pyrimidine derivatives as ALK-5 inhibitors Novartis AG (CH) 2008-01-16 EP disclosed