SCHEMBL4766580

SCHEMBL4766580

CCOC(=O)c1ccc(N(c2ccc(F)c(Cl)c2)[C@@H]2CCCN2C(=O)OC(C)(C)C)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.42
KMT2A Q03164 4/20 0.42
ALDH1A1 P00352 6/20 0.41
LMNA P02545 5/20 0.39
TSHR P16473 4/20 0.39
NPSR1 Q6W5P4 3/20 0.39
MAPT P10636 2/20 0.39
HTT P42858 2/20 0.39
MDM4 O15151 1/20 0.38
MDM2 Q00987 1/20 0.38
CETP P11597 2/20 0.38
TP53 P04637 1/20 0.37
POLB P06746 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
GAA P10253 2/20 0.37
NPC1 O15118 1/20 0.36
UCHL1 P09936 1/20 0.36
USP30 Q70CQ3 1/20 0.36
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4766576 1.00 MEN1 (0.42) MEN1KMT2AALDH1A1LMNATSHR
SCHEMBL4771661 0.88 ALDH1A1 (0.42) MEN1KMT2AALDH1A1LMNATSHR
SCHEMBL4771659 0.88 ALDH1A1 (0.42) MEN1KMT2AALDH1A1LMNATSHR
SCHEMBL4762739 0.86 ALDH1A1 (0.42) MEN1KMT2AALDH1A1LMNATSHR
SCHEMBL4762740 0.86 ALDH1A1 (0.42) MEN1KMT2AALDH1A1LMNATSHR
SCHEMBL330451 0.83 PGR (0.46) MEN1KMT2AALDH1A1LMNANPSR1
SCHEMBL330452 0.83 PGR (0.46) MEN1KMT2AALDH1A1LMNANPSR1
SCHEMBL4792059 0.83 ALDH1A1 (0.41) MEN1KMT2AALDH1A1LMNATSHR
SCHEMBL4792056 0.83 ALDH1A1 (0.41) MEN1KMT2AALDH1A1LMNATSHR
SCHEMBL4764121 0.83 APP (0.42) MEN1KMT2AALDH1A1LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881975-A1 N,N-SUBSTITUTED 3-AMINOPYRROLIDINE COMPOUNDS USEFUL AS MONOAMINES REUPTAKE INHIBITORS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-01-30 EP disclosed
WO-2006121218-A1 N,N-SUBSTITUTED 3-AMINOPYRROLIDINE COMPOUNDS USEFUL AS MONOAMINES REUPTAKE INHIBITORS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-11-16 WO disclosed