SCHEMBL4767283

SCHEMBL4767283

O=c1c([N+](=O)[O-])c(C=Cc2cnn(Cc3ccccc3F)c2)n(Cc2ccc(C(F)(F)F)cc2)c(=O)n1Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.35
ADORA2B P29275 3/20 0.35
ADORA1 P30542 3/20 0.35
MAPT P10636 3/20 0.35
ALDH1A1 P00352 2/20 0.35
PKM P14618 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KLKB1 P03952 1/20 0.34
HDAC2 Q92769 2/20 0.34
TGM2 P21980 1/20 0.33
P2RX3 P56373 1/20 0.33
TP53 P04637 1/20 0.33
GNRHR P30968 1/20 0.32
GAA P10253 1/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
KMT2A Q03164 1/20 0.32
TOP2A P11388 1/20 0.32
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4767273 1.00 ADORA2A (0.35) ADORA2AADORA2BADORA1MAPTALDH1A1
SCHEMBL4771562 0.93 ADORA2A (0.39) ADORA2AADORA2BADORA1ALDH1A1HDAC2
SCHEMBL4771574 0.93 ADORA2A (0.39) ADORA2AADORA2BADORA1ALDH1A1HDAC2
SCHEMBL4762591 0.91 MAPT (0.37) ADORA2AADORA2BADORA1MAPTALDH1A1
SCHEMBL4762596 0.91 MAPT (0.37) ADORA2AADORA2BADORA1MAPTALDH1A1
SCHEMBL4764053 0.90 ALDH1A1 (0.41) ADORA2AADORA2BADORA1MAPTALDH1A1
SCHEMBL4765667 0.89 ADORA2A (0.40) ADORA2AADORA2BADORA1MAPTALDH1A1
SCHEMBL4767816 0.88 MAPT (0.42) ADORA2AADORA2BADORA1MAPTALDH1A1
SCHEMBL4767823 0.88 MAPT (0.42) ADORA2AADORA2BADORA1MAPTALDH1A1
SCHEMBL4769234 0.87 NPBWR1 (0.41) ADORA2AADORA2BADORA1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678181-B1 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS INC (US) 2008-12-31 EP disclosed