SCHEMBL4771574

SCHEMBL4771574

O=c1c([N+](=O)[O-])c(C=Cc2cnn(Cc3ccccc3C(F)(F)F)c2)n(Cc2ccc(C(F)(F)F)cc2)c(=O)n1Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.39
ADORA2B P29275 3/20 0.39
ADORA1 P30542 3/20 0.39
ALDH1A1 P00352 1/20 0.35
MAPK1 P28482 1/20 0.35
SCD5 Q86SK9 1/20 0.34
TAS2R8 Q9NYW2 1/20 0.34
P2RX3 P56373 1/20 0.33
TGM2 P21980 1/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
KMT2A Q03164 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
NPBWR1 P48145 1/20 0.32
CYP2C8 P10632 2/20 0.32
CYP2B6 P20813 2/20 0.32
ADORA3 P0DMS8 1/20 0.32
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
HDAC2 Q92769 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4771562 1.00 ADORA2A (0.39) ADORA2AADORA2BADORA1ALDH1A1MAPK1
SCHEMBL4763418 0.93 ADORA2A (0.39) ADORA2AADORA2BADORA1ALDH1A1MAPK1
SCHEMBL4763420 0.93 ADORA2A (0.39) ADORA2AADORA2BADORA1ALDH1A1MAPK1
SCHEMBL4767273 0.93 ADORA2A (0.35) ADORA2AADORA2BADORA1ALDH1A1P2RX3
SCHEMBL4767283 0.93 ADORA2A (0.35) ADORA2AADORA2BADORA1ALDH1A1P2RX3
SCHEMBL4762462 0.91 NPBWR1 (0.44) ADORA2AADORA2BADORA1ALDH1A1MAPK1
SCHEMBL4762538 0.91 NPBWR1 (0.44) ADORA2AADORA2BADORA1ALDH1A1MAPK1
SCHEMBL4765667 0.88 ADORA2A (0.40) ADORA2AADORA2BADORA1ALDH1A1MAPK1
SCHEMBL4767385 0.88 ADORA2B (0.38) ADORA2AADORA2BADORA1ALDH1A1MAPK1
SCHEMBL4767375 0.88 ADORA2B (0.38) ADORA2AADORA2BADORA1ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678181-B1 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS INC (US) 2008-12-31 EP disclosed