SCHEMBL4767337

SCHEMBL4767337

[CH2]C[C@H](C)CC(=O)N(C1CCCNCC1=O)S(=O)(=O)c1ccccc1C#N

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
HTT P42858 1/20 0.35
HSD11B1 P28845 1/20 0.35
LMNA P02545 1/20 0.34
ATM Q13315 1/20 0.33
RORC P51449 1/20 0.33
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
BDKRB1 P46663 1/20 0.32
HCRTR2 O43614 1/20 0.31
KDM4E B2RXH2 1/20 0.30
NR1H3 Q13133 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4762038 0.91 ALDH1A1 (0.35) ALDH1A1HTTHSD11B1LMNAATM
SCHEMBL6637139 0.85 LMNA (0.32) ALDH1A1HTTHSD11B1LMNA
SCHEMBL7426348 0.82 ALDH1A1 (0.36) ALDH1A1HTTHSD11B1LMNAATM
SCHEMBL4907052 0.81
SCHEMBL6592307 0.81 PSEN1 (0.33)
SCHEMBL4766702 0.79 PSEN1 (0.41)
SCHEMBL7427475 0.79 PSEN1 (0.38) ALDH1A1
SCHEMBL7536966 0.79 ALDH1A1 (0.34) ALDH1A1HTTHSD11B1LMNAATM
SCHEMBL7434329 0.78 KCNA5 (0.35) HTTHSD11B1RORCSLC6A2SLC6A4
SCHEMBL6590952 0.78

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP claimed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP claimed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO claimed
EP-1320370-A4 METHOD OF TREATMENT SMITHKLINE BEECHAM CORP (US) 2008-10-22 EP disclosed
EP-1320370-A1 METHOD OF TREATMENT SmithKline Beecham Corporation (US) 2003-06-25 EP disclosed
WO-2002017924-A1 METHOD OF TREATMENT SMITHKLINE BEECHAM CORPORATION (GB) 2002-03-07 WO disclosed