SCHEMBL7426348

SCHEMBL7426348

CC(C)C[CH]C(=O)N([C@H]1CCCNCC1=O)S(=O)(=O)c1ccccc1C#N

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.36
HTT P42858 1/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
HSD11B1 P28845 1/20 0.35
LMNA P02545 1/20 0.34
ATM Q13315 1/20 0.34
RORC P51449 1/20 0.33
BDKRB1 P46663 1/20 0.31
KDM4E B2RXH2 1/20 0.31
NR1H3 Q13133 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30
HCRTR2 O43614 1/20 0.30
NOS1 P29475 3/20 0.30
NOS2 P35228 3/20 0.30
POLB P06746 1/20 0.30
GPR183 P32249 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7536966 0.92 ALDH1A1 (0.34) ALDH1A1HTTSLC6A2SLC6A4HSD11B1
SCHEMBL7433037 0.84
SCHEMBL4767337 0.82 ALDH1A1 (0.35) ALDH1A1HTTSLC6A2SLC6A4HSD11B1
SCHEMBL4907047 0.81
SCHEMBL4762038 0.81 ALDH1A1 (0.35) ALDH1A1HTTSLC6A2SLC6A4HSD11B1
SCHEMBL4761916 0.80 PSEN1 (0.33)
SCHEMBL6637135 0.80 SLC6A2 (0.35) ALDH1A1HTTSLC6A2SLC6A4HSD11B1
SCHEMBL4762983 0.80 PSEN1 (0.36) ALDH1A1LMNANR1H3
SCHEMBL7424733 0.79 PSEN1 (0.44)
SCHEMBL6591177 0.79 CTSK (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP claimed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP claimed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO claimed